Compile Data Set for Download or QSAR
maximum 50k data
Found 11 Enz. Inhib. hit(s) with all data for entry = 50020854
TargetCannabinoid receptor 2(Homo sapiens (Human))
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50218270((Z)-N-(5-tert-butyl-3-(cyclopropylmethyl)-4-methyl...)
Affinity DataIC50:  16nMAssay Description:Displacement of [3H] CP-55,940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50218272((Z)-N-(5-tert-butyl-3-(cyclopropylmethyl)-4-methyl...)
Affinity DataIC50:  65nMAssay Description:Displacement of [3H] CP-55,940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50218271((Z)-N-(3-allyl-5-tert-butyl-4-methylthiazol-2(3H)-...)
Affinity DataIC50:  75nMAssay Description:Displacement of [3H] CP-55,940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50218273((Z)-N-(5-tert-butyl-4-methyl-3-(3-methylbut-2-enyl...)
Affinity DataIC50:  170nMAssay Description:Displacement of [3H] CP-55,940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50218274((Z)-N-(5-tert-butyl-4-methyl-3-(prop-2-ynyl)thiazo...)
Affinity DataIC50:  210nMAssay Description:Displacement of [3H] CP-55,940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM5035(CHEMBL235747 | N-(5-tert-Butyl-3,4-dimethyl-1,3-th...)
Affinity DataIC50:  340nMAssay Description:Displacement of [3H] CP-55,940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50218275((Z)-N-(5-tert-butyl-3-(cyclopropylmethyl)-4-methyl...)
Affinity DataIC50:  490nMAssay Description:Displacement of [3H] CP-55,940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50218270((Z)-N-(5-tert-butyl-3-(cyclopropylmethyl)-4-methyl...)
Affinity DataIC50:  1.70E+3nMAssay Description:Displacement of [3H] CP-55,940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM5035(CHEMBL235747 | N-(5-tert-Butyl-3,4-dimethyl-1,3-th...)
Affinity DataIC50: >5.00E+4nMAssay Description:Displacement of [3H] CP-55,940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM5035(CHEMBL235747 | N-(5-tert-Butyl-3,4-dimethyl-1,3-th...)
Affinity DataEC50:  110nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells by [35S]GTPgamaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50218270((Z)-N-(5-tert-butyl-3-(cyclopropylmethyl)-4-methyl...)
Affinity DataEC50:  7.20nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells by [35S]GTPgamaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed