Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for entry = 50021356
TargetKappa-type opioid receptor(Homo sapiens (Human))
Holden Laboratories

Curated by ChEMBL
LigandPNGBDBM50223620(1-alpha-mesyloxysalvinorin A | CHEMBL439569)
Affinity DataEC50:  2.70E+3nMAssay Description:Agonist activity at human kappa opioid receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Holden Laboratories

Curated by ChEMBL
LigandPNGBDBM50159163((3S,4aR,4bS,6R,8R,8aR,10aR)-6-Acetoxy-3-furan-3-yl...)
Affinity DataEC50:  280nMAssay Description:Agonist activity at human kappa opioid receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Holden Laboratories

Curated by ChEMBL
LigandPNGBDBM50159165((2S,4aR,6aR,7R,9S,10aS,10bR)-9-(acetyloxy)-2-(fura...)
Affinity DataEC50:  1.24nMAssay Description:Agonist activity at human kappa opioid receptor assessed as inhibition of Galpha16-induced calcium fluxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Holden Laboratories

Curated by ChEMBL
LigandPNGBDBM50159163((3S,4aR,4bS,6R,8R,8aR,10aR)-6-Acetoxy-3-furan-3-yl...)
Affinity DataEC50:  3.34nMAssay Description:Agonist activity at human kappa opioid receptor assessed as inhibition of Galpha16-induced calcium fluxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed