Found 49 Enz. Inhib. hit(s) with all data for entry = 50038240 
Affinity DataKi: 1nMAssay Description:Displacement of [125I]NDP-MSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Displacement of [125I]NDP-MSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Displacement of [125I]NDP-MSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [125I]NDP-MSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Displacement of [125I]NDP-MSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Displacement of [125I]NDP-MSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Displacement of [125I]NDP-MSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Displacement of [125I]NDP-MSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Displacement of [125I]NDP-MSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.30nMAssay Description:Displacement of [125I]NDP-MSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.30nMAssay Description:Displacement of [125I]NDP-MSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.20nMAssay Description:Displacement of [125I]NDP-MSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.30nMAssay Description:Displacement of [125I]NDP-MSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.5nMAssay Description:Displacement of [125I]NDP-MSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.60nMAssay Description:Displacement of [125I]NDP-MSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [125I]NDP-MSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 51nMAssay Description:Displacement of [125I]NDP-MSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 61nMAssay Description:Displacement of [125I]NDP-MSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 90nMAssay Description:Displacement of [125I]NDP-MSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 120nMAssay Description:Binding affinity to MC1RMore data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Displacement of [125I]NDP-MSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:Binding affinity to MC3RMore data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:Displacement of [125I]NDP-MSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 290nMAssay Description:Displacement of [125I]NDP-MSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 370nMAssay Description:Displacement of [125I]NDP-MSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 470nMAssay Description:Displacement of [125I]NDP-MSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 530nMAssay Description:Binding affinity to MC5RMore data for this Ligand-Target Pair
Affinity DataKi: 560nMAssay Description:Displacement of [125I]NDP-MSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 800nMAssay Description:Binding affinity to MC5RMore data for this Ligand-Target Pair
Affinity DataKi: 850nMAssay Description:Displacement of [125I]NDP-MSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.30E+3nMAssay Description:Binding affinity to MC3RMore data for this Ligand-Target Pair
Affinity DataKi: 2.05E+3nMAssay Description:Displacement of [125I]NDP-MSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.70E+3nMAssay Description:Displacement of [125I]NDP-MSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.80E+3nMAssay Description:Displacement of [125I]NDP-MSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 64nMAssay Description:Antagonist activity at human MC4 receptor expressed in CHO cells assessed as inhibition of alpha-MSH-stimulated cAMP productionMore data for this Ligand-Target Pair
Affinity DataIC50: 560nMAssay Description:Antagonist activity at human MC4 receptor expressed in CHO cells assessed as inhibition of alpha-MSH-stimulated cAMP productionMore data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Agonist activity at human MC4 receptor expressed in CHO cells assessed as accumulation of cAMP productionMore data for this Ligand-Target Pair
Affinity DataEC50: 27nMAssay Description:Agonist activity at human MC4 receptor expressed in CHO cells assessed as accumulation of cAMP productionMore data for this Ligand-Target Pair
Affinity DataEC50: 19nMAssay Description:Agonist activity at human MC4 receptor expressed in CHO cells assessed as accumulation of cAMP productionMore data for this Ligand-Target Pair
Affinity DataEC50: 410nMAssay Description:Agonist activity at human MC4 receptor expressed in CHO cells assessed as accumulation of cAMP productionMore data for this Ligand-Target Pair
Affinity DataEC50: 79nMAssay Description:Agonist activity at human MC4 receptor expressed in CHO cells assessed as accumulation of cAMP productionMore data for this Ligand-Target Pair
Affinity DataEC50: 340nMAssay Description:Agonist activity at human MC4 receptor expressed in CHO cells assessed as accumulation of cAMP productionMore data for this Ligand-Target Pair
Affinity DataEC50: 44nMAssay Description:Agonist activity at human MC4 receptor expressed in CHO cells assessed as accumulation of cAMP productionMore data for this Ligand-Target Pair
Affinity DataEC50: 17nMAssay Description:Agonist activity at human MC4 receptor expressed in CHO cells assessed as accumulation of cAMP productionMore data for this Ligand-Target Pair
Affinity DataEC50: 16nMAssay Description:Agonist activity at human MC4 receptor expressed in CHO cells assessed as accumulation of cAMP productionMore data for this Ligand-Target Pair
Affinity DataEC50: 9.10nMAssay Description:Agonist activity at human MC4 receptor expressed in CHO cells assessed as accumulation of cAMP productionMore data for this Ligand-Target Pair
Affinity DataEC50: 10nMAssay Description:Agonist activity at human MC4 receptor expressed in CHO cells assessed as accumulation of cAMP productionMore data for this Ligand-Target Pair
Affinity DataEC50: 6nMAssay Description:Agonist activity at human MC4 receptor expressed in CHO cells assessed as accumulation of cAMP productionMore data for this Ligand-Target Pair
Affinity DataEC50: 5.20nMAssay Description:Agonist activity at human MC4 receptor expressed in CHO cells assessed as accumulation of cAMP productionMore data for this Ligand-Target Pair
