Compile Data Set for Download or QSAR
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Found 6 Enz. Inhib. hit(s) with all data for entry = 4976
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Research Institute, Hospital For Sick Children

LigandPNGBDBM84610(5-(3,5-dichlorophenoxy)-N-(4-pyrdinyl)-2- furamide...)
Affinity DataIC50:  4.70E+3nMpH: 5.5 T: 2°CAssay Description:Beta-glucocerebrosidase (GCase) activity was measured by release of 4-methylumbelliferyl fluorophore from MUClc.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Research Institute, Hospital For Sick Children

LigandPNGBDBM18046(5-((4-methylphenyl)thio)-quinazoline 2,4-diamine, ...)
Affinity DataIC50:  7.80E+3nMpH: 5.5 T: 2°CAssay Description:Beta-glucocerebrosidase (GCase) activity was measured by release of 4-methylumbelliferyl fluorophore from MUClc.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Research Institute, Hospital For Sick Children

LigandPNGBDBM84609(7,8-diethoxy-quinazoline 2,4-diamine, 1b)
Affinity DataIC50:  2.20E+4nMpH: 5.5 T: 2°CAssay Description:Beta-glucocerebrosidase (GCase) activity was measured by release of 4-methylumbelliferyl fluorophore from MUClc.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Research Institute, Hospital For Sick Children

LigandPNGBDBM84608(2,4-diamino-6-nitro-quinazoline, 1a)
Affinity DataIC50:  6.10E+4nMpH: 5.5 T: 2°CAssay Description:Beta-glucocerebrosidase (GCase) activity was measured by release of 4-methylumbelliferyl fluorophore from MUClc.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Research Institute, Hospital For Sick Children

LigandPNGBDBM84611(2-methyl-N-pyridin-4-yl-benzamide, 2a)
Affinity DataIC50:  8.00E+4nMpH: 5.5 T: 2°CAssay Description:Beta-glucocerebrosidase (GCase) activity was measured by release of 4-methylumbelliferyl fluorophore from MUClc.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Research Institute, Hospital For Sick Children

LigandPNGBDBM84612(2,2-dimethyl-N-(4-pyridinyl)propanamide, 2b)
Affinity DataIC50: >4.00E+5nMpH: 5.5 T: 2°CAssay Description:Beta-glucocerebrosidase (GCase) activity was measured by release of 4-methylumbelliferyl fluorophore from MUClc.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed