Compile Data Set for Download or QSAR
maximum 50k data
Found 46 Enz. Inhib. hit(s) with all data for entry = 50028007
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255312(2-(5-((dimethylamino)methyl)-2-methoxyphenyl)-4-(4...)
Affinity DataIC50:  6nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50239328(2-(3-((dimethylamino)methyl)phenyl)-4-(4-methyl-1H...)
Affinity DataIC50:  7.5nMAssay Description:Inhibition of human full length PKCthetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255312(2-(5-((dimethylamino)methyl)-2-methoxyphenyl)-4-(4...)
Affinity DataIC50:  8.70nMAssay Description:Inhibition of human full length PKCthetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255313(2-(5-((dimethylamino)methyl)-2-ethoxyphenyl)-4-(4-...)
Affinity DataIC50:  9.20nMAssay Description:Inhibition of human full length PKCthetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255315(2-(3-((dimethylamino)methyl)-2-methoxyphenyl)-4-(4...)
Affinity DataIC50:  12nMAssay Description:Inhibition of human full length PKCthetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50256031(2-(4-((dimethylamino)methyl)phenyl)-4-(4-methyl-1H...)
Affinity DataIC50:  14nMAssay Description:Inhibition of human full length PKCthetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255367(2-(2-((dimethylamino)methyl)-5-methoxyphenyl)-4-(4...)
Affinity DataIC50:  16nMAssay Description:Inhibition of human full length PKCthetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255252(2-(5-((dimethylamino)methyl)thiophen-3-yl)-4-(4-me...)
Affinity DataIC50:  16nMAssay Description:Inhibition of human full length PKCthetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255312(2-(5-((dimethylamino)methyl)-2-methoxyphenyl)-4-(4...)
Affinity DataIC50:  23nMAssay Description:Inhibition of LynMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255254(2-(2-methoxyphenyl)-4-(4-methyl-1H-indol-5-ylamino...)
Affinity DataIC50:  23nMAssay Description:Inhibition of human full length PKCthetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255312(2-(5-((dimethylamino)methyl)-2-methoxyphenyl)-4-(4...)
Affinity DataIC50:  24nMAssay Description:Inhibition of human full length PKCdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50239328(2-(3-((dimethylamino)methyl)phenyl)-4-(4-methyl-1H...)
Affinity DataIC50:  26nMAssay Description:Inhibition of human full length PKCdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255315(2-(3-((dimethylamino)methyl)-2-methoxyphenyl)-4-(4...)
Affinity DataIC50:  27nMAssay Description:Inhibition of human full length PKCdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50239328(2-(3-((dimethylamino)methyl)phenyl)-4-(4-methyl-1H...)
Affinity DataIC50:  28nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255252(2-(5-((dimethylamino)methyl)thiophen-3-yl)-4-(4-me...)
Affinity DataIC50:  51nMAssay Description:Inhibition of human full length PKCdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50239331(4-(1H-indol-5-ylamino)-2-phenylthieno[2,3-b]pyridi...)
Affinity DataIC50:  52nMAssay Description:Inhibition of human full length PKCthetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255313(2-(5-((dimethylamino)methyl)-2-ethoxyphenyl)-4-(4-...)
Affinity DataIC50:  74nMAssay Description:Inhibition of LynMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255313(2-(5-((dimethylamino)methyl)-2-ethoxyphenyl)-4-(4-...)
Affinity DataIC50:  82nMAssay Description:Inhibition of human full length PKCdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255253(2-(5-((dimethylamino)methyl)pyridin-3-yl)-4-(4-met...)
Affinity DataIC50:  84nMAssay Description:Inhibition of human full length PKCthetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50256031(2-(4-((dimethylamino)methyl)phenyl)-4-(4-methyl-1H...)
Affinity DataIC50:  88nMAssay Description:Inhibition of human full length PKCdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255251(2-(2-((dimethylamino)methyl)phenyl)-4-(4-methyl-1H...)
Affinity DataIC50:  93nMAssay Description:Inhibition of human full length PKCthetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50256031(2-(4-((dimethylamino)methyl)phenyl)-4-(4-methyl-1H...)
Affinity DataIC50:  100nMAssay Description:Inhibition of LynMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255314(2-(5-((dimethylamino)methyl)-2-methylphenyl)-4-(4-...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human full length PKCthetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255367(2-(2-((dimethylamino)methyl)-5-methoxyphenyl)-4-(4...)
Affinity DataIC50:  130nMAssay Description:Inhibition of human full length PKCdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255253(2-(5-((dimethylamino)methyl)pyridin-3-yl)-4-(4-met...)
Affinity DataIC50:  170nMAssay Description:Inhibition of human full length PKCdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255314(2-(5-((dimethylamino)methyl)-2-methylphenyl)-4-(4-...)
Affinity DataIC50:  230nMAssay Description:Inhibition of LynMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255254(2-(2-methoxyphenyl)-4-(4-methyl-1H-indol-5-ylamino...)
Affinity DataIC50:  250nMAssay Description:Inhibition of human full length PKCdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255254(2-(2-methoxyphenyl)-4-(4-methyl-1H-indol-5-ylamino...)
Affinity DataIC50:  310nMAssay Description:Inhibition of LynMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50239331(4-(1H-indol-5-ylamino)-2-phenylthieno[2,3-b]pyridi...)
Affinity DataIC50:  370nMAssay Description:Inhibition of human full length PKCdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255251(2-(2-((dimethylamino)methyl)phenyl)-4-(4-methyl-1H...)
Affinity DataIC50:  380nMAssay Description:Inhibition of human full length PKCdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255314(2-(5-((dimethylamino)methyl)-2-methylphenyl)-4-(4-...)
Affinity DataIC50:  410nMAssay Description:Inhibition of human full length PKCdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255252(2-(5-((dimethylamino)methyl)thiophen-3-yl)-4-(4-me...)
Affinity DataIC50:  410nMAssay Description:Inhibition of LynMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50239328(2-(3-((dimethylamino)methyl)phenyl)-4-(4-methyl-1H...)
Affinity DataIC50:  520nMAssay Description:Inhibition of LynMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255315(2-(3-((dimethylamino)methyl)-2-methoxyphenyl)-4-(4...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of LynMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255253(2-(5-((dimethylamino)methyl)pyridin-3-yl)-4-(4-met...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of LynMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50239331(4-(1H-indol-5-ylamino)-2-phenylthieno[2,3-b]pyridi...)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of LynMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase HCK(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255367(2-(2-((dimethylamino)methyl)-5-methoxyphenyl)-4-(4...)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of HckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255367(2-(2-((dimethylamino)methyl)-5-methoxyphenyl)-4-(4...)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of FynMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-activated protein kinase 2(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255367(2-(2-((dimethylamino)methyl)-5-methoxyphenyl)-4-(4...)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255367(2-(2-((dimethylamino)methyl)-5-methoxyphenyl)-4-(4...)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255367(2-(2-((dimethylamino)methyl)-5-methoxyphenyl)-4-(4...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of LynMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255367(2-(2-((dimethylamino)methyl)-5-methoxyphenyl)-4-(4...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of human full length PKCbetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255251(2-(2-((dimethylamino)methyl)phenyl)-4-(4-methyl-1H...)
Affinity DataIC50:  3.70E+4nMAssay Description:Inhibition of LynMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255367(2-(2-((dimethylamino)methyl)-5-methoxyphenyl)-4-(4...)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255367(2-(2-((dimethylamino)methyl)-5-methoxyphenyl)-4-(4...)
Affinity DataIC50:  9.50E+4nMAssay Description:Inhibition of human full length PKCepsilonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255367(2-(2-((dimethylamino)methyl)-5-methoxyphenyl)-4-(4...)
Affinity DataIC50:  3.60E+5nMAssay Description:Inhibition of human full length PKCetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed