Compile Data Set for Download or QSAR
maximum 50k data
Found 94 Enz. Inhib. hit(s) with all data for entry = 50028172
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248651(2,4-dichloro-N-((4-(6-methylpyridin-2-yl)-1-(propy...)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248641(2-amino-6-chloro-N-((4-phenyl-1-(propylsulfonyl)pi...)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of glycine transporter 1 (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248058((S)-2,4-dichloro-N-(1-(1-(propylsulfonyl)-4-(pyrid...)
Affinity DataIC50:  3nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248669(2-chloro-N-((4-(6-methylpyridin-2-yl)-1-(propylsul...)
Affinity DataIC50:  3nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248667(2,4-dichloro-N-((4-(4-methylpyridin-2-yl)-1-(propy...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248059((S)-2-chloro-3,5-difluoro-N-(1-(1-(propylsulfonyl)...)
Affinity DataIC50:  4nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248100((2,4-dichloro-N-((1-(propylsulfonyl)-4-(pyridin-2-...)
Affinity DataIC50:  4.40nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248648(3,6-dichloro-2-fluoro-N-((1-(propylsulfonyl)-4-(py...)
Affinity DataIC50:  5.70nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248646(2,6-dichloro-N-((1-(propylsulfonyl)-4-(pyridin-2-y...)
Affinity DataIC50:  6.60nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248647(2-amino-6-chloro-N-((1-(propylsulfonyl)-4-(pyridin...)
Affinity DataIC50:  6.90nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248653(2-chloro-N-((4-(6-methoxypyridin-2-yl)-1-(propylsu...)
Affinity DataIC50:  6.90nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248670(2,4-dichloro-N-((4-(6-methoxypyridin-2-yl)-1-(prop...)
Affinity DataIC50:  7.40nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248125(2,4-dichloro-N-((1-methyl-1'-(propylsulfonyl)-2,4'...)
Affinity DataIC50:  9.5nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248681(2-chloro-N-((1-(propylsulfonyl)-4-(pyridin-2-yl)pi...)
Affinity DataIC50:  12nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248013((S)-N-(1-(1-(propylsulfonyl)-4-(pyridin-2-yl)piper...)
Affinity DataIC50:  18nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248665(CHEMBL517034 | N-((1-(propylsulfonyl)-4-(pyridin-2...)
Affinity DataIC50:  19nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248644(2-methyl-N-((1-(propylsulfonyl)-4-(pyridin-2-yl)pi...)
Affinity DataIC50:  20nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248094(CHEMBL460922 | N-((1-methyl-1'-(propylsulfonyl)-2,...)
Affinity DataIC50:  21nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248664(CHEMBL465426 | N-((1-(propylsulfonyl)-4-(pyridin-2...)
Affinity DataIC50:  31nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248666(2-chloro-N-((4-(4-methylpyridin-2-yl)-1-(propylsul...)
Affinity DataIC50:  38nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248126(2-chloro-3,5-difluoro-N-((1-methyl-1'-(propylsulfo...)
Affinity DataIC50:  43nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248652(CHEMBL465129 | N-((4-(6-methoxypyridin-2-yl)-1-(pr...)
Affinity DataIC50:  48nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248643(2-fluoro-N-((1-(propylsulfonyl)-4-(pyridin-2-yl)pi...)
Affinity DataIC50:  49nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248668(CHEMBL463238 | N-((4-(6-methylpyridin-2-yl)-1-(pro...)
Affinity DataIC50:  55nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248095(2-chloro-N-((1-methyl-1'-(propylsulfonyl)-2,4'-bip...)
Affinity DataIC50:  59nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248060(2,4-dichloro-N-((1-(propylsulfonyl)-4-(pyridin-3-y...)
Affinity DataIC50:  69nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248061(2,4-dichloro-N-((1-(propylsulfonyl)-4-(pyridin-4-y...)
Affinity DataIC50:  79nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248682(4-chloro-N-((1-(propylsulfonyl)-4-(pyridin-2-yl)pi...)
Affinity DataIC50:  103nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248642(CHEMBL518686 | N-((1-(propylsulfonyl)-4-(pyridin-2...)
Affinity DataIC50:  107nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248649(CHEMBL517631 | N-((4-(4-methylpyridin-2-yl)-1-(pro...)
Affinity DataIC50:  129nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248680(2-methoxy-N-((4-phenyl-1-(propylsulfonyl)piperidin...)
Affinity DataIC50:  130nMAssay Description:Inhibition of glycine transporter 1 (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248684(3,4-dichloro-N-((1-(propylsulfonyl)-4-(pyridin-2-y...)
Affinity DataIC50:  131nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248093(2-methyl-N-((1-methyl-1'-(propylsulfonyl)-2,4'-bip...)
Affinity DataIC50:  148nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248673(2,4-dichloro-N-((4-(6-morpholinopyridin-2-yl)-1-(p...)
Affinity DataIC50:  412nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248672(2-chloro-N-((4-(6-morpholinopyridin-2-yl)-1-(propy...)
Affinity DataIC50:  482nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248683(3-chloro-N-((1-(propylsulfonyl)-4-(pyridin-2-yl)pi...)
Affinity DataIC50:  517nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248012((R)-2-chloro-3,5-difluoro-N-(1-(1-(propylsulfonyl)...)
Affinity DataIC50:  576nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248011((R)-2,4-dichloro-N-(1-(1-(propylsulfonyl)-4-(pyrid...)
Affinity DataIC50:  661nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248663(3-methyl-N-((1-(propylsulfonyl)-4-(pyridin-2-yl)pi...)
Affinity DataIC50:  833nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248010((R)-N-(1-(1-(propylsulfonyl)-4-(pyridin-2-yl)piper...)
Affinity DataIC50:  2.59E+3nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248092(CHEMBL518339 | N-((1-methyl-1'-(propylsulfonyl)-2,...)
Affinity DataIC50:  3.31E+3nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248671(CHEMBL463433 | N-((4-(6-morpholinopyridin-2-yl)-1-...)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of human glycine transporter 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248100((2,4-dichloro-N-((1-(propylsulfonyl)-4-(pyridin-2-...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of glycine transporter 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248684(3,4-dichloro-N-((1-(propylsulfonyl)-4-(pyridin-2-y...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of glycine transporter 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248648(3,6-dichloro-2-fluoro-N-((1-(propylsulfonyl)-4-(py...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of glycine transporter 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248647(2-amino-6-chloro-N-((1-(propylsulfonyl)-4-(pyridin...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of glycine transporter 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248649(CHEMBL517631 | N-((4-(4-methylpyridin-2-yl)-1-(pro...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of glycine transporter 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248644(2-methyl-N-((1-(propylsulfonyl)-4-(pyridin-2-yl)pi...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of glycine transporter 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248681(2-chloro-N-((1-(propylsulfonyl)-4-(pyridin-2-yl)pi...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of glycine transporter 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50248643(2-fluoro-N-((1-(propylsulfonyl)-4-(pyridin-2-yl)pi...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of glycine transporter 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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