Compile Data Set for Download or QSAR
maximum 50k data
Found 72 Enz. Inhib. hit(s) with all data for entry = 50030272
TargetProstaglandin E2 receptor EP4 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM35847((15S)-prostaglandin E2 | (5Z,11alpha,13E,15S)-11,1...)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of rat EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP2 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM35847((15S)-prostaglandin E2 | (5Z,11alpha,13E,15S)-11,1...)
Affinity DataIC50:  5.20nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293496(2-(3-((N-(4-tert-butylbenzyl)pyridine-3-sulfonamid...)
Affinity DataIC50:  50nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293493(3-(3-((N-(4-tert-butylbenzyl)pyridine-2-sulfonamid...)
Affinity DataIC50:  52nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293495(3-(3-((N-(4-tert-butylbenzyl)thiazole-2-sulfonamid...)
Affinity DataIC50:  63nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293498(7-(N-(4-(1-hydroxyhexyl)benzyl)methylsulfonamido)h...)
Affinity DataIC50:  93nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293502(7-(N-(4-butylbenzyl)methylsulfonamido)heptanoic ac...)
Affinity DataIC50:  160nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293497(7-(N-(4-hydroxynonyl)methylsulfonamido)heptanoic a...)
Affinity DataIC50:  225nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293490(3-(3-((N-(4-butylbenzyl)methylsulfonamido)methyl)p...)
Affinity DataIC50:  270nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293492(3-(3-((N-(4-tert-butylbenzyl)phenylsulfonamido)met...)
Affinity DataIC50:  278nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293503(7-(N-(biphenyl-4-ylmethyl)methylsulfonamido)heptan...)
Affinity DataIC50:  289nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293494(2-(3-((N-(4-tert-butylbenzyl)-1-(1-methyl-1H-imida...)
Affinity DataIC50:  326nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293491(3-(3-((N-(4-tert-butylbenzyl)methylsulfonamido)met...)
Affinity DataIC50:  379nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293509(4-(2-(N-(4-butylbenzyl)methylsulfonamido)phenyl)bu...)
Affinity DataIC50:  494nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293501(7-(N-(4-(1-hydroxypentyl)benzyl)methylsulfonamido)...)
Affinity DataIC50:  502nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293504(7-(N-(4-tert-butylbenzyl)methylsulfonamido)heptano...)
Affinity DataIC50:  590nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293500(7-(N-(4-hexanoylbenzyl)methylsulfonamido)heptanoic...)
Affinity DataIC50:  636nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293510(4-(4-(N-(4-butylbenzyl)methylsulfonamido)phenyl)bu...)
Affinity DataIC50:  654nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293505(2-(4-(N-(4-butylbenzyl)methylsulfonamido)butoxy)ac...)
Affinity DataIC50:  701nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293489(2-(3-((N-(4-tert-butylbenzyl)methylsulfonamido)met...)
Affinity DataIC50:  792nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293507(2-(4-(2-(N-(4-butylbenzyl)methylsulfonamido)ethyl)...)
Affinity DataIC50:  833nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293488(6-(N-(4-hydroxynonyl)methylsulfonamido)hexanoic ac...)
Affinity DataIC50:  910nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293504(7-(N-(4-tert-butylbenzyl)methylsulfonamido)heptano...)
Affinity DataIC50:  2.47E+3nMAssay Description:Inhibition of rat EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293499(7-(N-(4-hydroxy-6-methylheptyl)methylsulfonamido)h...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293497(7-(N-(4-hydroxynonyl)methylsulfonamido)heptanoic a...)
Affinity DataIC50:  2.53E+3nMAssay Description:Inhibition of rat EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293506(3-(3-(N-(4-butylbenzyl)methylsulfonamido)propoxy)b...)
Affinity DataIC50:  3.13E+3nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293498(7-(N-(4-(1-hydroxyhexyl)benzyl)methylsulfonamido)h...)
Affinity DataIC50: >3.20E+3nMAssay Description:Inhibition of rat EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293499(7-(N-(4-hydroxy-6-methylheptyl)methylsulfonamido)h...)
Affinity DataIC50: >3.20E+3nMAssay Description:Inhibition of rat EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293500(7-(N-(4-hexanoylbenzyl)methylsulfonamido)heptanoic...)
Affinity DataIC50: >3.20E+3nMAssay Description:Inhibition of rat EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293501(7-(N-(4-(1-hydroxypentyl)benzyl)methylsulfonamido)...)
Affinity DataIC50: >3.20E+3nMAssay Description:Inhibition of rat EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293502(7-(N-(4-butylbenzyl)methylsulfonamido)heptanoic ac...)
Affinity DataIC50: >3.20E+3nMAssay Description:Inhibition of rat EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293503(7-(N-(biphenyl-4-ylmethyl)methylsulfonamido)heptan...)
Affinity DataIC50: >3.20E+3nMAssay Description:Inhibition of rat EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293511(3-(3-(N-(4-butylbenzyl)methylsulfonamido)phenyl)pr...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293506(3-(3-(N-(4-butylbenzyl)methylsulfonamido)propoxy)b...)
Affinity DataIC50: >3.20E+3nMAssay Description:Inhibition of rat EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293507(2-(4-(2-(N-(4-butylbenzyl)methylsulfonamido)ethyl)...)
Affinity DataIC50: >3.20E+3nMAssay Description:Inhibition of rat EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293508(2-(2-((N-(4-butylbenzyl)methylsulfonamido)methyl)p...)
Affinity DataIC50: >3.20E+3nMAssay Description:Inhibition of rat EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293509(4-(2-(N-(4-butylbenzyl)methylsulfonamido)phenyl)bu...)
Affinity DataIC50: >3.20E+3nMAssay Description:Inhibition of rat EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293510(4-(4-(N-(4-butylbenzyl)methylsulfonamido)phenyl)bu...)
Affinity DataIC50: >3.20E+3nMAssay Description:Inhibition of rat EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293511(3-(3-(N-(4-butylbenzyl)methylsulfonamido)phenyl)pr...)
Affinity DataIC50: >3.20E+3nMAssay Description:Inhibition of rat EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293489(2-(3-((N-(4-tert-butylbenzyl)methylsulfonamido)met...)
Affinity DataIC50: >3.20E+3nMAssay Description:Inhibition of rat EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293490(3-(3-((N-(4-butylbenzyl)methylsulfonamido)methyl)p...)
Affinity DataIC50: >3.20E+3nMAssay Description:Inhibition of rat EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293491(3-(3-((N-(4-tert-butylbenzyl)methylsulfonamido)met...)
Affinity DataIC50: >3.20E+3nMAssay Description:Inhibition of rat EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293492(3-(3-((N-(4-tert-butylbenzyl)phenylsulfonamido)met...)
Affinity DataIC50: >3.20E+3nMAssay Description:Inhibition of rat EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293493(3-(3-((N-(4-tert-butylbenzyl)pyridine-2-sulfonamid...)
Affinity DataIC50: >3.20E+3nMAssay Description:Inhibition of rat EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293494(2-(3-((N-(4-tert-butylbenzyl)-1-(1-methyl-1H-imida...)
Affinity DataIC50: >3.20E+3nMAssay Description:Inhibition of rat EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293512(3-(3-((N-(4-tert-butylbenzyl)-4-chlorophenylsulfon...)
Affinity DataIC50: >3.20E+3nMAssay Description:Inhibition of rat EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293495(3-(3-((N-(4-tert-butylbenzyl)thiazole-2-sulfonamid...)
Affinity DataIC50: >3.20E+3nMAssay Description:Inhibition of rat EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293487(5-(N-(4-hydroxynonyl)methylsulfonamido)pentanoic a...)
Affinity DataIC50: >3.20E+3nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293496(2-(3-((N-(4-tert-butylbenzyl)pyridine-3-sulfonamid...)
Affinity DataIC50: >3.20E+3nMAssay Description:Inhibition of rat EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50293512(3-(3-((N-(4-tert-butylbenzyl)-4-chlorophenylsulfon...)
Affinity DataIC50: >3.20E+3nMAssay Description:Inhibition of rat EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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