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Found 6 Enz. Inhib. hit(s) with all data for entry = 50032919
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50336510(7,8-dihydroxy-1-methoxy-3-methyl-10-oxo-1,10-dihyd...)
Affinity DataKi:  180nMAssay Description:Inhibition of Pseudomonas aeruginosa beta-lactamase IMP-1 assessed as hydrolysis of nitrocefin by UV spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50336511((4R,5S,6S)-3-(benzo[b]thiophen-2-ylthio)-6-((R)-1-...)
Affinity DataKi:  180nMAssay Description:Inhibition of Pseudomonas aeruginosa beta-lactamase IMP-1 assessed as hydrolysis of nitrocefin by UV spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50336509(CHEMBL116455 | Mercapto-acetic acid | Mercaptoacet...)
Affinity DataKi:  180nMAssay Description:Inhibition of Pseudomonas aeruginosa beta-lactamase IMP-1 assessed as hydrolysis of nitrocefin by UV spectrophotometric analysisMore data for this Ligand-Target Pair
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50121953(2-mercaptoethanecarboxylic acid | 3-mercaptopropan...)
Affinity DataKi:  180nMAssay Description:Inhibition of Pseudomonas aeruginosa beta-lactamase IMP-1 assessed as hydrolysis of nitrocefin by UV spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50336508(CHEMBL1673299 | sodium 2,3-diethylmaleate)
Affinity DataKi:  410nMAssay Description:Inhibition of Pseudomonas aeruginosa beta-lactamase IMP-1 assessed as hydrolysis of nitrocefin by UV spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase VIM-2(Pseudomonas aeruginosa (g-Proteobacteria))
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50336508(CHEMBL1673299 | sodium 2,3-diethylmaleate)
Affinity DataKi:  1.20E+5nMAssay Description:Inhibition of Pseudomonas aeruginosa beta-lactamase VIM-2 assessed as hydrolysis of nitrocefin by UV spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed