Compile Data Set for Download or QSAR
maximum 50k data
Found 26 Enz. Inhib. hit(s) with all data for entry = 50032197
TargetVasopressin V1b receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325847(CHEMBL1223814 | N-(cyclopropylmethyl)-2-(6-(3-morp...)
Affinity DataIC50:  120nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325825((S)-2-amino-N-((S)-1-(3-(2-(cyclopropylmethylamino...)
Affinity DataIC50:  200nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(RAT)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325847(CHEMBL1223814 | N-(cyclopropylmethyl)-2-(6-(3-morp...)
Affinity DataIC50:  210nMAssay Description:Displacement of [3H]AVP from rat vasopressin V3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325842(CHEMBL1223699 | N-(cyclopropylmethyl)-2-(4-oxo-2-p...)
Affinity DataIC50:  310nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325844(2-(6-(3-(azepan-1-yl)propoxy)-4-oxo-2-phenylquinaz...)
Affinity DataIC50:  340nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325845(CHEMBL1223757 | N-(cyclopropylmethyl)-2-(6-(3-(4-m...)
Affinity DataIC50:  710nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325846(CHEMBL1223758 | N-(cyclopropylmethyl)-2-(6-(3-(4-h...)
Affinity DataIC50:  1.10E+3nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325837(CHEMBL1223632 | N-(cyclopropylmethyl)-2-(6-(3-(4-m...)
Affinity DataIC50:  1.70E+3nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325843(CHEMBL1223755 | N-(cyclopropylmethyl)-2-(4-oxo-2-p...)
Affinity DataIC50:  1.80E+3nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325830((S)-2-(6-(2-amino-4-methylpentyloxy)-4-oxo-2-pheny...)
Affinity DataIC50:  2.10E+3nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325832(2-(6-(3-aminopropoxy)-4-oxo-2-phenylquinazolin-3(4...)
Affinity DataIC50:  3.60E+3nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325841(CHEMBL1223698 | N-(cyclopropylmethyl)-2-(6-(3-(die...)
Affinity DataIC50:  3.80E+3nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325831(2-(6-(2-aminoethoxy)-4-oxo-2-phenylquinazolin-3(4H...)
Affinity DataIC50:  4.00E+3nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325838(CHEMBL1223633 | N-(cyclopropylmethyl)-2-(6-(4-(4-m...)
Affinity DataIC50:  4.80E+3nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325826((S)-2-amino-N-(1-(3-(2-(cyclopropylmethylamino)-2-...)
Affinity DataIC50:  5.10E+3nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325840(CHEMBL1223697 | N-(cyclopropylmethyl)-2-(6-(3-(met...)
Affinity DataIC50:  7.60E+3nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325836(CHEMBL1223631 | N-(cyclopropylmethyl)-2-(6-(2-(4-m...)
Affinity DataIC50:  2.20E+4nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325839(CHEMBL1223696 | N-(cyclopropylmethyl)-2-(4-oxo-2-p...)
Affinity DataIC50:  2.58E+4nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325834(2-(6-(5-aminopentyloxy)-4-oxo-2-phenylquinazolin-3...)
Affinity DataIC50: >3.00E+4nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325833(2-(6-(4-aminobutoxy)-4-oxo-2-phenylquinazolin-3(4H...)
Affinity DataIC50: >3.00E+4nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325827(2-amino-N-(2-(3-(2-(cyclopropylmethylamino)-2-oxoe...)
Affinity DataIC50:  3.05E+4nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325847(CHEMBL1223814 | N-(cyclopropylmethyl)-2-(6-(3-morp...)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of [3H]AVP from human vasopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325847(CHEMBL1223814 | N-(cyclopropylmethyl)-2-(6-(3-morp...)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of [3H]oxytocin from human oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325828(CHEMBL1224609 | N-(2-(3-(2-(cyclopropylmethylamino...)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325835(2-(6-(6-aminohexyloxy)-4-oxo-2-phenylquinazolin-3(...)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50325829(CHEMBL1224610 | N-(cyclopropylmethyl)-2-(6-hydroxy...)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of [3H]AVP from human vasopresin3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed