TargetATP-binding cassette sub-family C member 3(Homo sapiens (Human))
University Hospital Heidelberg
Curated by ChEMBL
University Hospital Heidelberg
Curated by ChEMBL
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of MRP3 expressed in MDCK2 cells assessed as cell growth inhibition by calcein and pheophorbide A efflux assaysMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
University Hospital Heidelberg
Curated by ChEMBL
University Hospital Heidelberg
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of BCRP expressed in MDCK2 cells assessed as cell growth inhibition by calcein and pheophorbide A efflux assaysMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
University Hospital Heidelberg
Curated by ChEMBL
University Hospital Heidelberg
Curated by ChEMBL
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibition of MDR1 expressed in MDCK2 cells assessed as inhibition of cell proliferation by calcein and pheophorbide A efflux assaysMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 2(Homo sapiens (Human))
University Hospital Heidelberg
Curated by ChEMBL
University Hospital Heidelberg
Curated by ChEMBL
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibition of MRP2 expressed in MDCK2 cells assessed as cell growth inhibition by calcein and pheophorbide A efflux assaysMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
University Hospital Heidelberg
Curated by ChEMBL
University Hospital Heidelberg
Curated by ChEMBL
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibition of MRP1 expressed in MDCK2 cells assessed as cell growth inhibition by calcein and pheophorbide A efflux assaysMore data for this Ligand-Target Pair