TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Caprotec Bioanalytics
Curated by ChEMBL
Caprotec Bioanalytics
Curated by ChEMBL
Affinity DataKi: 900nMAssay Description:Inhibition of human recombinant NQO2-mediated mitomycin C metabolism using NADH as cosubstrate incubated for 5 mins prior to NADH addition measured a...More data for this Ligand-Target Pair
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Caprotec Bioanalytics
Curated by ChEMBL
Caprotec Bioanalytics
Curated by ChEMBL
Affinity DataKi: 6.00E+4nMAssay Description:Inhibition of human recombinant NQO2-mediated mitomycin C metabolism using NADH as cosubstrate incubated for 5 mins prior to NADH addition measured a...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of human thrombin-mediated platelet aggregation in cell-based assayMore data for this Ligand-Target Pair
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Caprotec Bioanalytics
Curated by ChEMBL
Caprotec Bioanalytics
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Competitive inhibition of human recombinant NQO2-mediated mitomycin C metabolism using NADH as cosubstrate incubated for 5 mins prior to NADH additio...More data for this Ligand-Target Pair
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Caprotec Bioanalytics
Curated by ChEMBL
Caprotec Bioanalytics
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Competitive inhibition of human recombinant NQO2-mediated mitomycin C metabolism using NADH as cosubstrate incubated for 5 mins prior to NADH additio...More data for this Ligand-Target Pair
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Caprotec Bioanalytics
Curated by ChEMBL
Caprotec Bioanalytics
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Displacement of (S)-N4-(4-(3-(2-((4-carbamimidoylphenylamino)methyl)-1-methyl-N-(pyridin-2-yl)-1H-benzo[d]imidazole-5-carboxamido)propanamido)butyl)-...More data for this Ligand-Target Pair
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Caprotec Bioanalytics
Curated by ChEMBL
Caprotec Bioanalytics
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Competitive inhibition of human recombinant NQO2-mediated mitomycin C metabolism using NADH as cosubstrate incubated for 5 mins prior to NADH additio...More data for this Ligand-Target Pair
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Caprotec Bioanalytics
Curated by ChEMBL
Caprotec Bioanalytics
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Displacement of (S)-N4-(4-(3-(2-((4-carbamimidoylphenylamino)methyl)-1-methyl-N-(pyridin-2-yl)-1H-benzo[d]imidazole-5-carboxamido)propanamido)butyl)-...More data for this Ligand-Target Pair