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Found 4 Enz. Inhib. hit(s) with all data for entry = 50042974
TargetMitogen-activated protein kinase 7(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50434072(CHEMBL2381342)
Affinity DataIC50:  59nMAssay Description:Inhibition of ERK5 phosphorylation in sorbitol-stimulated human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 7(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50434071(CHEMBL2381341)
Affinity DataIC50:  810nMAssay Description:Inhibition of ERK5 phosphorylation in sorbitol-stimulated human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 7(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50434069(CHEMBL2381339 | US9676792, Compound 24)
Affinity DataEC50: >3.00E+4nMAssay Description:Inhibition of GST-tagged full length human ERK5 transfected in HEK293 cells assessed as inhibition of AP1 transcriptional activity after 24 hrs by du...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 7(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50434070(CHEMBL2381340)
Affinity DataEC50:  4.20E+3nMAssay Description:Inhibition of GST-tagged full length human ERK5 transfected in HEK293 cells assessed as inhibition of AP1 transcriptional activity after 24 hrs by du...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed