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Found 4 Enz. Inhib. hit(s) with all data for entry = 7990
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM227598(Penem 1)
Affinity DataKi:  30nM IC50:  150nMpH: 7.2Assay Description:Steady-state kinetics were performed on an Agilent 8453 diode array spectrophotometer (Palo Alto, CA) in 50 mM sodium phosphate buffer (pH 7.2) suppl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase OXA-1(Escherichia coli (Enterobacteria))
Case Western Reserve University

LigandPNGBDBM227598(Penem 1)
Affinity DataKi:  50nM IC50:  30nMpH: 7.2Assay Description:Steady-state kinetics were performed on an Agilent 8453 diode array spectrophotometer (Palo Alto, CA) in 50 mM sodium phosphate buffer (pH 7.2) suppl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM227599(Penem 3)
Affinity DataKi:  150nM IC50:  160nMpH: 7.2Assay Description:Steady-state kinetics were performed on an Agilent 8453 diode array spectrophotometer (Palo Alto, CA) in 50 mM sodium phosphate buffer (pH 7.2) suppl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase OXA-1(Escherichia coli (Enterobacteria))
Case Western Reserve University

LigandPNGBDBM227599(Penem 3)
Affinity DataKi:  380nM IC50:  60nMpH: 7.2Assay Description:Steady-state kinetics were performed on an Agilent 8453 diode array spectrophotometer (Palo Alto, CA) in 50 mM sodium phosphate buffer (pH 7.2) suppl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed