TargetRecQ-like DNA helicase BLM(Homo sapiens (Human))
Drexel University College Of Medicine
Curated by ChEMBL
Drexel University College Of Medicine
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of BLM helicase (unknown origin) binding to DNAMore data for this Ligand-Target Pair
TargetBifunctional 3'-5' exonuclease/ATP-dependent helicase WRN(Homo sapiens (Human))
Drexel University College Of Medicine
Curated by ChEMBL
Drexel University College Of Medicine
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of WRN helicase (unknown origin)More data for this Ligand-Target Pair
TargetDouble-strand break repair protein MRE11(Homo sapiens (Human))
Drexel University College Of Medicine
Curated by ChEMBL
Drexel University College Of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.20E+4nMAssay Description:In vitro inhibition of purified recombinant Mre11 exonuclease activity (unknown origin)More data for this Ligand-Target Pair
TargetBifunctional 3'-5' exonuclease/ATP-dependent helicase WRN(Homo sapiens (Human))
Drexel University College Of Medicine
Curated by ChEMBL
Drexel University College Of Medicine
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of WRN helicase (unknown origin)More data for this Ligand-Target Pair
TargetRecQ-like DNA helicase BLM(Homo sapiens (Human))
Drexel University College Of Medicine
Curated by ChEMBL
Drexel University College Of Medicine
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of BLM helicase (unknown origin) assessed as branch migration activityMore data for this Ligand-Target Pair
TargetDouble-strand break repair protein MRE11(Homo sapiens (Human))
Drexel University College Of Medicine
Curated by ChEMBL
Drexel University College Of Medicine
Curated by ChEMBL
Affinity DataIC50: 6.60E+4nMAssay Description:Inhibition of Mre11 exonuclease activity (unknown origin) in cell free extractsMore data for this Ligand-Target Pair
TargetDNA repair and recombination protein RAD54-like(Homo sapiens (Human))
Drexel University College Of Medicine
Curated by ChEMBL
Drexel University College Of Medicine
Curated by ChEMBL
Affinity DataEC50: 1.65E+4nMAssay Description:Inhibition of RAD54 (unknown origin) ATPase activity assessed as generation of reactive oxygen speciesMore data for this Ligand-Target Pair
TargetCell cycle checkpoint protein RAD1(Homo sapiens (Human))
Drexel University College Of Medicine
Curated by ChEMBL
Drexel University College Of Medicine
Curated by ChEMBL
Affinity DataEC50: 4.40E+4nMAssay Description:Inhibition of RAD1 (unknown origin) binding to ssDNAMore data for this Ligand-Target Pair
TargetCell cycle checkpoint protein RAD1(Homo sapiens (Human))
Drexel University College Of Medicine
Curated by ChEMBL
Drexel University College Of Medicine
Curated by ChEMBL
Affinity DataEC50: 1.00E+3nMAssay Description:Inhibition of RAD1 (unknown origin) binding to ssDNAMore data for this Ligand-Target Pair
TargetCell cycle checkpoint protein RAD1(Homo sapiens (Human))
Drexel University College Of Medicine
Curated by ChEMBL
Drexel University College Of Medicine
Curated by ChEMBL
Affinity DataKd: 2.00E+3nMAssay Description:Binding affinity to RAD1 (unknown origin) by surface plasmon resonance methodMore data for this Ligand-Target Pair
TargetCell cycle checkpoint protein RAD1(Homo sapiens (Human))
Drexel University College Of Medicine
Curated by ChEMBL
Drexel University College Of Medicine
Curated by ChEMBL
Affinity DataEC50: 5.00E+3nMAssay Description:Inhibition of RAD1 (unknown origin) binding to ssDNAMore data for this Ligand-Target Pair
TargetCell cycle checkpoint protein RAD1(Homo sapiens (Human))
Drexel University College Of Medicine
Curated by ChEMBL
Drexel University College Of Medicine
Curated by ChEMBL
Affinity DataKd: 5.60E+3nMAssay Description:Binding affinity to RAD1 (unknown origin) by surface plasmon resonance methodMore data for this Ligand-Target Pair
TargetCell cycle checkpoint protein RAD1(Homo sapiens (Human))
Drexel University College Of Medicine
Curated by ChEMBL
Drexel University College Of Medicine
Curated by ChEMBL
Affinity DataEC50: 2.70E+4nMAssay Description:Inhibition of RAD1 (unknown origin) binding to ssDNAMore data for this Ligand-Target Pair