Compile Data Set for Download or QSAR
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Found 19 Enz. Inhib. hit(s) with all data for entry = 50044783
TargetSortase family protein(Staphylococcus aureus)
University Of Latvia

Curated by ChEMBL
LigandPNGBDBM50030337(CHEMBL3343843)
Affinity DataIC50:  3.39E+3nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSortase family protein(Staphylococcus aureus)
University Of Latvia

Curated by ChEMBL
LigandPNGBDBM50030335(CHEMBL3343842)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSortase family protein(Staphylococcus aureus)
University Of Latvia

Curated by ChEMBL
LigandPNGBDBM50030322(CHEMBL3343832)
Affinity DataIC50:  3.81E+3nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSortase family protein(Staphylococcus aureus)
University Of Latvia

Curated by ChEMBL
LigandPNGBDBM50030321(CHEMBL3343831)
Affinity DataIC50:  3.87E+3nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSortase family protein(Staphylococcus aureus)
University Of Latvia

Curated by ChEMBL
LigandPNGBDBM50030329(CHEMBL3343839)
Affinity DataIC50:  3.96E+3nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSortase family protein(Staphylococcus aureus)
University Of Latvia

Curated by ChEMBL
LigandPNGBDBM50030327(CHEMBL3343837)
Affinity DataIC50:  4.01E+3nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSortase family protein(Staphylococcus aureus)
University Of Latvia

Curated by ChEMBL
LigandPNGBDBM50030328(CHEMBL3343838)
Affinity DataIC50:  4.07E+3nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSortase family protein(Staphylococcus aureus)
University Of Latvia

Curated by ChEMBL
LigandPNGBDBM50030336(CHEMBL3341779)
Affinity DataIC50:  4.22E+3nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSortase family protein(Staphylococcus aureus)
University Of Latvia

Curated by ChEMBL
LigandPNGBDBM50030323(CHEMBL3343833)
Affinity DataIC50:  4.62E+3nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSortase family protein(Staphylococcus aureus)
University Of Latvia

Curated by ChEMBL
LigandPNGBDBM50030320(CHEMBL3343830)
Affinity DataIC50:  4.99E+3nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSortase family protein(Staphylococcus aureus)
University Of Latvia

Curated by ChEMBL
LigandPNGBDBM50030334(CHEMBL3343841)
Affinity DataIC50:  5.06E+3nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSortase family protein(Staphylococcus aureus)
University Of Latvia

Curated by ChEMBL
LigandPNGBDBM50030326(CHEMBL3343836)
Affinity DataIC50:  5.08E+3nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSortase family protein(Staphylococcus aureus)
University Of Latvia

Curated by ChEMBL
LigandPNGBDBM34709(MLS000567780 | N-(1-adamantyl)-2-(3-keto-1,2-benzo...)
Affinity DataIC50:  6.11E+3nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSortase family protein(Staphylococcus aureus)
University Of Latvia

Curated by ChEMBL
LigandPNGBDBM50030330(CHEMBL3343840)
Affinity DataIC50:  6.26E+3nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSortase family protein(Staphylococcus aureus)
University Of Latvia

Curated by ChEMBL
LigandPNGBDBM50030325(CHEMBL3343835)
Affinity DataIC50:  6.44E+3nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSortase family protein(Staphylococcus aureus)
University Of Latvia

Curated by ChEMBL
LigandPNGBDBM50030324(CHEMBL3343834)
Affinity DataIC50:  7.06E+3nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSortase family protein(Staphylococcus aureus)
University Of Latvia

Curated by ChEMBL
LigandPNGBDBM50030338(CHEMBL3343844)
Affinity DataIC50:  1.28E+4nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSortase family protein(Staphylococcus aureus)
University Of Latvia

Curated by ChEMBL
LigandPNGBDBM50201782(1-(3,4-dichlorophenyl)-3-(dimethylamino)propan-1-o...)
Affinity DataIC50:  1.69E+4nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSortase family protein(Staphylococcus aureus)
University Of Latvia

Curated by ChEMBL
LigandPNGBDBM50125084((ethenylsulfonyl)benzene | CHEMBL165058 | Ethenesu...)
Affinity DataIC50:  7.36E+5nMAssay Description:Inhibition of Staphylococcus aureus sortase A using dabcyl-QALPETGEE-edans as substrate incubated for 1 hr prior to substrate addition measured at 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed