BindingDB PrimarySearch_ki

Found 25 Enz. Inhib. hit(s) with all data for entry = 50045615

Protein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia

Curated by ChEMBL

PNG

BDBM50009672(AdoHcy | CHEMBL418052 | S-(5'-adenosyl)-L-homocyst...)

IC50: 420nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair

PDB
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3D Structure (crystal)

Protein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia

Curated by ChEMBL

PNG

BDBM50070953(CHEMBL3409550)

IC50: 610nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
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CHEMBL PC cid PC sid Similars

Details Article PubMed

Protein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia

Curated by ChEMBL

PNG

BDBM50071013(CHEMBL3409546)

IC50: 1.15E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
B.MOAD GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Protein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia

Curated by ChEMBL

PNG

BDBM50071012(CHEMBL3409549)

IC50: 1.25E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
B.MOAD GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Protein arginine N-methyltransferase 5(Homo sapiens (Human))
The University Of Georgia

Curated by ChEMBL

PNG

BDBM50070953(CHEMBL3409550)

IC50: 1.40E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT5 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Protein arginine N-methyltransferase 8(Homo sapiens (Human))
The University Of Georgia

Curated by ChEMBL

PNG

BDBM50070953(CHEMBL3409550)

IC50: 1.74E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT8 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Protein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia

Curated by ChEMBL

PNG

BDBM50070954(CHEMBL3099810)

IC50: 1.81E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
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CHEMBL PC cid PC sid Similars

Details Article PubMed

Protein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia

Curated by ChEMBL

PNG

BDBM50070952(CHEMBL3409555)

IC50: 2.03E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
B.MOAD GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Protein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia

Curated by ChEMBL

PNG

BDBM50070957(CHEMBL3409561)

IC50: 2.37E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
B.MOAD GoogleScholar

CHEMBL PC cid PC sid Patents Similars

Details Article PubMed

Protein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia

Curated by ChEMBL

PNG

BDBM50387486(CHEMBL2047486)

IC50: 2.56E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
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Details Article PubMed

Protein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia

Curated by ChEMBL

PNG

BDBM50071010(CHEMBL3409554)

IC50: 2.67E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
B.MOAD GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Protein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia

Curated by ChEMBL

PNG

BDBM50070951(CHEMBL3409558)

IC50: 3.05E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
B.MOAD GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Protein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia

Curated by ChEMBL

PNG

BDBM50070950(CHEMBL3409562)

IC50: 3.38E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
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CHEMBL PC cid PC sid Similars

Details Article PubMed

Protein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia

Curated by ChEMBL

PNG

BDBM50070956(CHEMBL3409563)

IC50: 3.39E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
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Details Article PubMed

Protein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia

Curated by ChEMBL

PNG

BDBM50070958(CHEMBL3409557)

IC50: 4.00E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
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CHEMBL PC cid PC sid Similars

Details Article PubMed

Protein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia

Curated by ChEMBL

PNG

BDBM50070955(CHEMBL3409565)

IC50: 5.76E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
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CHEMBL PC cid PC sid Patents Similars

Details Article PubMed

Histone-arginine methyltransferase CARM1(Homo sapiens (Human))
The University Of Georgia

Curated by ChEMBL

PNG

BDBM50070951(CHEMBL3409558)

IC50: 5.80E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged CARM1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Protein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia

Curated by ChEMBL

PNG

BDBM50071011(CHEMBL3409553)

IC50: 6.43E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
B.MOAD GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Protein arginine N-methyltransferase 5(Homo sapiens (Human))
The University Of Georgia

Curated by ChEMBL

PNG

BDBM50070951(CHEMBL3409558)

IC50: 7.04E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT5 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Histone-arginine methyltransferase CARM1(Homo sapiens (Human))
The University Of Georgia

Curated by ChEMBL

PNG

BDBM50070952(CHEMBL3409555)

IC50: 7.23E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged CARM1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Protein arginine N-methyltransferase 5(Homo sapiens (Human))
The University Of Georgia

Curated by ChEMBL

PNG

BDBM50070952(CHEMBL3409555)

IC50: 8.36E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT5 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Histone-arginine methyltransferase CARM1(Homo sapiens (Human))
The University Of Georgia

Curated by ChEMBL

PNG

BDBM50070950(CHEMBL3409562)

IC50: 2.15E+4nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged CARM1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Protein arginine N-methyltransferase 8(Homo sapiens (Human))
The University Of Georgia

Curated by ChEMBL

PNG

BDBM50070951(CHEMBL3409558)

IC50: 2.84E+4nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT8 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Protein arginine N-methyltransferase 5(Homo sapiens (Human))
The University Of Georgia

Curated by ChEMBL

PNG

BDBM50070950(CHEMBL3409562)

IC50: 3.54E+4nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT5 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Protein arginine N-methyltransferase 8(Homo sapiens (Human))
The University Of Georgia

Curated by ChEMBL

PNG

BDBM50070950(CHEMBL3409562)

IC50: 8.49E+4nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT8 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed