Compile Data Set for Download or QSAR
maximum 50k data
Found 69 Enz. Inhib. hit(s) with all data for entry = 4754
TargetNorepinephrine transporter(RAT)
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM81946(CAS_96850-13-4 | LU 19,005 | LU 19-005)
Affinity DataKi:  0.260nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM81946(CAS_96850-13-4 | LU 19,005 | LU 19-005)
Affinity DataKi:  0.480nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM50021895(4-(3,4-Dichloro-phenyl)-7-methoxy-2-methyl-1,2,3,4...)
Affinity DataKi:  0.740nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNorepinephrine transporter(RAT)
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM50021217(CHEMBL52247 | Talsupram | [3-(3,3-Dimethyl-1-pheny...)
Affinity DataKi:  0.790nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM81946(CAS_96850-13-4 | LU 19,005 | LU 19-005)
Affinity DataKi:  0.990nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM25870(1-[3-(dimethylamino)propyl]-1-(4-fluorophenyl)-1,3...)
Affinity DataKi:  1.80nMMore data for this Ligand-Target Pair
TargetNorepinephrine transporter(RAT)
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM50021895(4-(3,4-Dichloro-phenyl)-7-methoxy-2-methyl-1,2,3,4...)
Affinity DataKi:  2.30nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM81954(1-(2-Benzhydryloxy-ethyl)-4-((E)-3-phenyl-allyl)-p...)
Affinity DataKi:  2.60nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNorepinephrine transporter(RAT)
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM22417(3-(2-methoxyphenoxy)-N-methyl-3-phenylpropan-1-ami...)
Affinity DataKi:  3.40nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM50021895(4-(3,4-Dichloro-phenyl)-7-methoxy-2-methyl-1,2,3,4...)
Affinity DataKi:  3.70nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM22199(1-{2-[bis(4-fluorophenyl)methoxy]ethyl}-4-[(2E)-3-...)
In DepthDetails ArticlePubMed
TargetNorepinephrine transporter(RAT)
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM50026952((cis) [3-(3,4-Dichloro-phenyl)-bicyclo[2.2.2]oct-2...)
Affinity DataKi:  5.40nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNorepinephrine transporter(RAT)
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM50005548((+)-2-Methyl-4-phenyl-1,2,3,4-tetrahydro-isoquinol...)
Affinity DataKi:  6.60nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM50026952((cis) [3-(3,4-Dichloro-phenyl)-bicyclo[2.2.2]oct-2...)
Affinity DataKi:  9.30nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNorepinephrine transporter(RAT)
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM22199(1-{2-[bis(4-fluorophenyl)methoxy]ethyl}-4-[(2E)-3-...)
Affinity DataKi:  13nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNorepinephrine transporter(RAT)
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM81954(1-(2-Benzhydryloxy-ethyl)-4-((E)-3-phenyl-allyl)-p...)
Affinity DataKi:  29nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM50005548((+)-2-Methyl-4-phenyl-1,2,3,4-tetrahydro-isoquinol...)
Affinity DataKi:  48nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM50026952((cis) [3-(3,4-Dichloro-phenyl)-bicyclo[2.2.2]oct-2...)
Affinity DataKi:  51nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM22199(1-{2-[bis(4-fluorophenyl)methoxy]ethyl}-4-[(2E)-3-...)
Affinity DataKi:  74nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM81954(1-(2-Benzhydryloxy-ethyl)-4-((E)-3-phenyl-allyl)-p...)
Affinity DataKi:  270nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM81946(CAS_96850-13-4 | LU 19,005 | LU 19-005)
Affinity DataKi:  290nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM50021895(4-(3,4-Dichloro-phenyl)-7-methoxy-2-methyl-1,2,3,4...)
Affinity DataKi:  480nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM50021895(4-(3,4-Dichloro-phenyl)-7-methoxy-2-methyl-1,2,3,4...)
Affinity DataKi:  550nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM22417(3-(2-methoxyphenoxy)-N-methyl-3-phenylpropan-1-ami...)
Affinity DataKi:  560nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM50026952((cis) [3-(3,4-Dichloro-phenyl)-bicyclo[2.2.2]oct-2...)
Affinity DataKi:  570nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM50048392(2-(tert-butylamino)-1-(3-chlorophenyl)propan-1-one...)
Affinity DataKi:  600nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM22417(3-(2-methoxyphenoxy)-N-methyl-3-phenylpropan-1-ami...)
Affinity DataKi:  610nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM22417(3-(2-methoxyphenoxy)-N-methyl-3-phenylpropan-1-ami...)
Affinity DataKi:  620nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM81946(CAS_96850-13-4 | LU 19,005 | LU 19-005)
Affinity DataKi:  740nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM22199(1-{2-[bis(4-fluorophenyl)methoxy]ethyl}-4-[(2E)-3-...)
Affinity DataKi:  810nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM50005548((+)-2-Methyl-4-phenyl-1,2,3,4-tetrahydro-isoquinol...)
Affinity DataKi:  830nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM50021217(CHEMBL52247 | Talsupram | [3-(3,3-Dimethyl-1-pheny...)
Affinity DataKi:  850nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM81954(1-(2-Benzhydryloxy-ethyl)-4-((E)-3-phenyl-allyl)-p...)
Affinity DataKi:  900nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM81954(1-(2-Benzhydryloxy-ethyl)-4-((E)-3-phenyl-allyl)-p...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM50005548((+)-2-Methyl-4-phenyl-1,2,3,4-tetrahydro-isoquinol...)
Affinity DataKi:  1.20E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50021217(CHEMBL52247 | Talsupram | [3-(3,3-Dimethyl-1-pheny...)
Affinity DataKi:  1.30E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNorepinephrine transporter(RAT)
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM50048392(2-(tert-butylamino)-1-(3-chlorophenyl)propan-1-one...)
Affinity DataKi:  1.50E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM25870(1-[3-(dimethylamino)propyl]-1-(4-fluorophenyl)-1,3...)
Affinity DataKi:  1.60E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM50021217(CHEMBL52247 | Talsupram | [3-(3,3-Dimethyl-1-pheny...)
Affinity DataKi:  1.60E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM81954(1-(2-Benzhydryloxy-ethyl)-4-((E)-3-phenyl-allyl)-p...)
Affinity DataKi:  1.90E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM22199(1-{2-[bis(4-fluorophenyl)methoxy]ethyl}-4-[(2E)-3-...)
Affinity DataKi:  2.20E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM22199(1-{2-[bis(4-fluorophenyl)methoxy]ethyl}-4-[(2E)-3-...)
Affinity DataKi:  2.20E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM81954(1-(2-Benzhydryloxy-ethyl)-4-((E)-3-phenyl-allyl)-p...)
Affinity DataKi:  2.50E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM22199(1-{2-[bis(4-fluorophenyl)methoxy]ethyl}-4-[(2E)-3-...)
Affinity DataKi:  3.40E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50021895(4-(3,4-Dichloro-phenyl)-7-methoxy-2-methyl-1,2,3,4...)
Affinity DataKi:  3.70E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM50005548((+)-2-Methyl-4-phenyl-1,2,3,4-tetrahydro-isoquinol...)
Affinity DataKi:  3.80E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM22417(3-(2-methoxyphenoxy)-N-methyl-3-phenylpropan-1-ami...)
Affinity DataKi:  4.30E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM25870(1-[3-(dimethylamino)propyl]-1-(4-fluorophenyl)-1,3...)
Affinity DataKi:  4.80E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM22417(3-(2-methoxyphenoxy)-N-methyl-3-phenylpropan-1-ami...)
Affinity DataKi:  5.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNorepinephrine transporter(RAT)
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM25870(1-[3-(dimethylamino)propyl]-1-(4-fluorophenyl)-1,3...)
Affinity DataKi:  8.80E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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