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Found 76 Enz. Inhib. hit(s) with all data for entry = 50035447
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50029150(3-(2-Piperidin-4-yl-ethyl)-1H-indole | CHEMBL27652...)
Affinity DataIC50:  10nMAssay Description:Inhibition of uptake of 5-HT in rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM77970(3-(2-chloranyl-5,6-dihydrobenzo[b][1]benzazepin-11...)
Affinity DataIC50:  20nMAssay Description:Inhibition of uptake of 5-HT in rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50029145(3-(2-Piperidin-4-yl-ethyl)-1H-indol-5-ol; fumarate)
Affinity DataIC50:  20nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50029150(3-(2-Piperidin-4-yl-ethyl)-1H-indole | CHEMBL27652...)
Affinity DataIC50:  30nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50029140(3-(3-Piperidin-4-yl-propyl)-1H-indole | CHEMBL2404...)
Affinity DataIC50:  40nMAssay Description:Inhibition of uptake of 5-HT in rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50029157(3-Piperidin-4-ylmethyl-1H-indole | CHEMBL429771)
Affinity DataIC50:  50nMAssay Description:Inhibition of uptake of 5-HT in rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50029140(3-(3-Piperidin-4-yl-propyl)-1H-indole | CHEMBL2404...)
Affinity DataIC50:  60nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM77970(3-(2-chloranyl-5,6-dihydrobenzo[b][1]benzazepin-11...)
Affinity DataIC50:  70nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50029154(5-Fluoro-3-piperidin-4-ylmethyl-1H-indole | CHEMBL...)
Affinity DataIC50:  100nMAssay Description:Inhibition of uptake of 5-HT in rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50029141(5-Chloro-3-(2-piperidin-4-yl-ethyl)-1H-indole | CH...)
Affinity DataIC50:  130nMAssay Description:Inhibition of uptake of 5-HT in rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50029153(5-Methoxy-3-(2-piperidin-4-yl-ethyl)-1H-indole | C...)
Affinity DataIC50:  140nMAssay Description:Inhibition of uptake of 5-HT in rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50029146(3-(2-Piperidin-4-yl-ethyl)-1H-indol-6-ol; fumarate)
Affinity DataIC50:  150nMAssay Description:Inhibition of uptake of dopamine (DA) rat brain striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50029154(5-Fluoro-3-piperidin-4-ylmethyl-1H-indole | CHEMBL...)
Affinity DataIC50:  170nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50029141(5-Chloro-3-(2-piperidin-4-yl-ethyl)-1H-indole | CH...)
Affinity DataIC50:  220nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50029151(1-Benzyl-3-(2-piperidin-4-yl-ethyl)-1H-indole; hyd...)
Affinity DataIC50:  300nMAssay Description:Inhibition of uptake of dopamine (DA) rat brain striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50029143(1-Methyl-3-(2-piperidin-4-yl-ethyl)-1H-indole; hyd...)
Affinity DataIC50:  400nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50029142(1-Phenyl-3-(2-piperidin-4-yl-ethyl)-1H-indole; fum...)
Affinity DataIC50:  400nMAssay Description:Inhibition of uptake of noradrenaline in rat brain hypothalamusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50029143(1-Methyl-3-(2-piperidin-4-yl-ethyl)-1H-indole; hyd...)
Affinity DataIC50:  400nMAssay Description:Inhibition of uptake of 5-HT in rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50029152(3-[2-(1-Methyl-piperidin-4-yl)-ethyl]-1H-indole | ...)
Affinity DataIC50:  450nMAssay Description:Inhibition of uptake of 5-HT in rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50029140(3-(3-Piperidin-4-yl-propyl)-1H-indole | CHEMBL2404...)
Affinity DataIC50:  500nMAssay Description:Inhibition of uptake of noradrenaline in rat brain hypothalamusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50029157(3-Piperidin-4-ylmethyl-1H-indole | CHEMBL429771)
Affinity DataIC50:  550nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50029145(3-(2-Piperidin-4-yl-ethyl)-1H-indol-5-ol; fumarate)
Affinity DataIC50:  600nMAssay Description:Inhibition of uptake of 5-HT in rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50029146(3-(2-Piperidin-4-yl-ethyl)-1H-indol-6-ol; fumarate)
Affinity DataIC50:  600nMAssay Description:Inhibition of uptake of noradrenaline in rat brain hypothalamusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50029148(5-Bromo-3-piperidin-4-ylmethyl-1H-indole | CHEMBL2...)
Affinity DataIC50:  600nMAssay Description:Inhibition of uptake of noradrenaline in rat brain hypothalamusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50029141(5-Chloro-3-(2-piperidin-4-yl-ethyl)-1H-indole | CH...)
Affinity DataIC50:  650nMAssay Description:Inhibition of uptake of noradrenaline in rat brain hypothalamusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50029148(5-Bromo-3-piperidin-4-ylmethyl-1H-indole | CHEMBL2...)
Affinity DataIC50:  700nMAssay Description:Inhibition of uptake of 5-HT in rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM77970(3-(2-chloranyl-5,6-dihydrobenzo[b][1]benzazepin-11...)
Affinity DataIC50:  700nMAssay Description:Inhibition of uptake of noradrenaline in rat brain hypothalamusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50029144(5-Chloro-3-piperidin-4-ylmethyl-1H-indole; 5 moles...)
Affinity DataIC50:  700nMAssay Description:Inhibition of uptake of 5-HT in rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50029142(1-Phenyl-3-(2-piperidin-4-yl-ethyl)-1H-indole; fum...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of uptake of 5-HT in rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50029148(5-Bromo-3-piperidin-4-ylmethyl-1H-indole | CHEMBL2...)
Affinity DataIC50:  1.00E+3nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50029147(2-Phenyl-3-(2-piperidin-4-yl-ethyl)-1H-indole | CH...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50029146(3-(2-Piperidin-4-yl-ethyl)-1H-indol-6-ol; fumarate)
Affinity DataIC50: >1.00E+3nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50029155(5-Methoxy-3-piperidin-4-ylmethyl-1H-indole | CHEMB...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50029155(5-Methoxy-3-piperidin-4-ylmethyl-1H-indole | CHEMB...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of uptake of 5-HT in rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50029154(5-Fluoro-3-piperidin-4-ylmethyl-1H-indole | CHEMBL...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of uptake of noradrenaline in rat brain hypothalamusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50029152(3-[2-(1-Methyl-piperidin-4-yl)-ethyl]-1H-indole | ...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50029153(5-Methoxy-3-(2-piperidin-4-yl-ethyl)-1H-indole | C...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50029144(5-Chloro-3-piperidin-4-ylmethyl-1H-indole; 5 moles...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50029156(1-Methyl-3-[2-(1-methyl-piperidin-4-yl)-ethyl]-1H-...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM77970(3-(2-chloranyl-5,6-dihydrobenzo[b][1]benzazepin-11...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of uptake of dopamine (DA) rat brain striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50029151(1-Benzyl-3-(2-piperidin-4-yl-ethyl)-1H-indole; hyd...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50029145(3-(2-Piperidin-4-yl-ethyl)-1H-indol-5-ol; fumarate)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of uptake of noradrenaline in rat brain hypothalamusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50029142(1-Phenyl-3-(2-piperidin-4-yl-ethyl)-1H-indole; fum...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50029149(2-Methyl-3-(2-piperidin-4-yl-ethyl)-1H-indole | CH...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50029143(1-Methyl-3-(2-piperidin-4-yl-ethyl)-1H-indole; hyd...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of uptake of noradrenaline in rat brain hypothalamusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50029141(5-Chloro-3-(2-piperidin-4-yl-ethyl)-1H-indole | CH...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of uptake of dopamine (DA) rat brain striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50029157(3-Piperidin-4-ylmethyl-1H-indole | CHEMBL429771)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of uptake of noradrenaline in rat brain hypothalamusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50029147(2-Phenyl-3-(2-piperidin-4-yl-ethyl)-1H-indole | CH...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of uptake of noradrenaline in rat brain hypothalamusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50029146(3-(2-Piperidin-4-yl-ethyl)-1H-indol-6-ol; fumarate)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of uptake of 5-HT in rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50029150(3-(2-Piperidin-4-yl-ethyl)-1H-indole | CHEMBL27652...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of uptake of noradrenaline in rat brain hypothalamusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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