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PubMed code 9784091

Compile data set for download or QSAR
Found 25 hits of Enzyme Inhibition Constant Data   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Cholinesterases


(Homo sapiens (Human))
BDBM50067482
PNG
(6-[(2-Methoxy-benzyl)-methyl-amino]-hexanoic acid ...)
Show SMILES COc1ccccc1CN(C)CCCCCC(=O)N(C)CCCCCCCCN(C)C(=O)CCCCCN(C)Cc1ccccc1OC
Show InChI InChI=1S/C40H66N4O4/c1-41(33-35-23-15-17-25-37(35)47-5)29-19-11-13-27-39(45)43(3)31-21-9-7-8-10-22-32-44(4)40(46)28-14-12-20-30-42(2)34-36-24-16-18-26-38(36)48-6/h15-18,23-26H,7-14,19-22,27-34H2,1-6H3
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0.100n/an/an/an/an/an/an/an/a



University of Bologna

Curated by ChEMBL


Assay Description
Inhibition constant determined against Acetylcholinesterase (AChE) receptor.


J Med Chem 41: 4186-9 (1998)

Checked by Author
Article DOI: 10.1021/jm9810452
BindingDB Entry DOI: 10.7270/Q2HH6KRM
More data for this
Ligand-Target Pair
Choline Acetyltransferase


(RAT)
BDBM8961
PNG
(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Show SMILES Nc1c2CCCCc2nc2ccccc12
Show InChI InChI=1S/C13H14N2/c14-13-9-5-1-3-7-11(9)15-12-8-4-2-6-10(12)13/h1,3,5,7H,2,4,6,8H2,(H2,14,15)
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0.150n/an/an/an/an/an/an/an/a



University of Bologna

Curated by ChEMBL


Assay Description
Inhibition constant determined against Acetylcholinesterase (AChE) receptor.


J Med Chem 41: 4186-9 (1998)

Checked by Author
Article DOI: 10.1021/jm9810452
BindingDB Entry DOI: 10.7270/Q2HH6KRM
More data for this
Ligand-Target Pair
Cholinesterases


(Homo sapiens (Human))
BDBM120262
PNG
(EDROPHONIUM BROMIDE | EDROPHONIUM CHLORIDE | Edrop...)
Show SMILES CC[N+](C)(C)c1cccc(O)c1
Show InChI InChI=1S/C10H15NO/c1-4-11(2,3)9-6-5-7-10(12)8-9/h5-8H,4H2,1-3H3/p+1
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1.60n/an/an/an/an/an/an/an/a



University of Bologna

Curated by ChEMBL


Assay Description
Inhibition constant determined against Acetylcholinesterase (AChE) receptor.


J Med Chem 41: 4186-9 (1998)

Checked by Author
Article DOI: 10.1021/jm9810452
BindingDB Entry DOI: 10.7270/Q2HH6KRM
More data for this
Ligand-Target Pair
Cholinesterases


(Homo sapiens (Human))
BDBM11023
PNG
((3aS,8aR)-1,3a,8-trimethyl-1H,2H,3H,3aH,8H,8aH-pyr...)
Show SMILES CNC(=O)Oc1ccc2N(C)[C@H]3N(C)CC[C@@]3(C)c2c1
Show InChI InChI=1/C15H21N3O2/c1-15-7-8-17(3)13(15)18(4)12-6-5-10(9-11(12)15)20-14(19)16-2/h5-6,9,13H,7-8H2,1-4H3,(H,16,19)/t13-,15+/s2
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n/an/a 14n/an/an/an/an/an/a



University of Bologna

Curated by ChEMBL


Assay Description
Inhibition of acetylcholinesterase (AChE) of human erythrocytes


J Med Chem 41: 4186-9 (1998)

Checked by Author
Article DOI: 10.1021/jm9810452
BindingDB Entry DOI: 10.7270/Q2HH6KRM
More data for this
Ligand-Target Pair
Cholinesterases


(Homo sapiens (Human))
BDBM11023
PNG
((3aS,8aR)-1,3a,8-trimethyl-1H,2H,3H,3aH,8H,8aH-pyr...)
Show SMILES CNC(=O)Oc1ccc2N(C)[C@H]3N(C)CC[C@@]3(C)c2c1
Show InChI InChI=1/C15H21N3O2/c1-15-7-8-17(3)13(15)18(4)12-6-5-10(9-11(12)15)20-14(19)16-2/h5-6,9,13H,7-8H2,1-4H3,(H,16,19)/t13-,15+/s2
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n/an/a 23n/an/an/an/an/an/a



University of Bologna

Curated by ChEMBL


Assay Description
Inhibition of Butyrylcholinesterase (BChE) of human erythrocytes [-log IC50 (uM)]


J Med Chem 41: 4186-9 (1998)

Checked by Author
Article DOI: 10.1021/jm9810452
BindingDB Entry DOI: 10.7270/Q2HH6KRM
More data for this
Ligand-Target Pair
Cholinesterases


(Homo sapiens (Human))
BDBM50067482
PNG
(6-[(2-Methoxy-benzyl)-methyl-amino]-hexanoic acid ...)
Show SMILES COc1ccccc1CN(C)CCCCCC(=O)N(C)CCCCCCCCN(C)C(=O)CCCCCN(C)Cc1ccccc1OC
Show InChI InChI=1S/C40H66N4O4/c1-41(33-35-23-15-17-25-37(35)47-5)29-19-11-13-27-39(45)43(3)31-21-9-7-8-10-22-32-44(4)40(46)28-14-12-20-30-42(2)34-36-24-16-18-26-38(36)48-6/h15-18,23-26H,7-14,19-22,27-34H2,1-6H3
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n/an/a 170n/an/an/an/an/an/a



University of Bologna

Curated by ChEMBL


Assay Description
Inhibition of acetylcholinesterase (AChE) of human erythrocytes


J Med Chem 41: 4186-9 (1998)

Checked by Author
Article DOI: 10.1021/jm9810452
BindingDB Entry DOI: 10.7270/Q2HH6KRM
More data for this
Ligand-Target Pair
Cholinesterases


(Homo sapiens (Human))
BDBM8961
PNG
(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Show SMILES Nc1c2CCCCc2nc2ccccc12
Show InChI InChI=1S/C13H14N2/c14-13-9-5-1-3-7-11(9)15-12-8-4-2-6-10(12)13/h1,3,5,7H,2,4,6,8H2,(H2,14,15)
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n/an/a 219n/an/an/an/an/an/a



University of Bologna

Curated by ChEMBL


Assay Description
Inhibition of acetylcholinesterase (AChE) of human erythrocytes


J Med Chem 41: 4186-9 (1998)

Checked by Author
Article DOI: 10.1021/jm9810452
BindingDB Entry DOI: 10.7270/Q2HH6KRM
More data for this
Ligand-Target Pair
Cholinesterases


(Homo sapiens (Human))
BDBM50422269
PNG
(CHEMBL132377)
Show SMILES COc1ccccc1CNCCCCCC(=O)N(C)CCCCCCCCN(C)C(=O)CCCCCNCc1ccccc1OC
Show InChI InChI=1S/C38H62N4O4/c1-41(37(43)25-11-9-17-27-39-31-33-21-13-15-23-35(33)45-3)29-19-7-5-6-8-20-30-42(2)38(44)26-12-10-18-28-40-32-34-22-14-16-24-36(34)46-4/h13-16,21-24,39-40H,5-12,17-20,25-32H2,1-4H3
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n/an/a 309n/an/an/an/an/an/a



University of Bologna

Curated by ChEMBL


Assay Description
Inhibition of acetylcholinesterase (AChE) of human erythrocytes


J Med Chem 41: 4186-9 (1998)

Checked by Author
Article DOI: 10.1021/jm9810452
BindingDB Entry DOI: 10.7270/Q2HH6KRM
More data for this
Ligand-Target Pair
Cholinesterases


(Homo sapiens (Human))
BDBM8961
PNG
(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Show SMILES Nc1c2CCCCc2nc2ccccc12
Show InChI InChI=1S/C13H14N2/c14-13-9-5-1-3-7-11(9)15-12-8-4-2-6-10(12)13/h1,3,5,7H,2,4,6,8H2,(H2,14,15)
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n/an/a 363n/an/an/an/an/an/a



University of Bologna

Curated by ChEMBL


Assay Description
Inhibition of Butyrylcholinesterase (BChE) of human erythrocytes [-log IC50 (uM)]


J Med Chem 41: 4186-9 (1998)

Checked by Author
Article DOI: 10.1021/jm9810452
BindingDB Entry DOI: 10.7270/Q2HH6KRM
More data for this
Ligand-Target Pair
3D
3D Structure (crystal)
Cholinesterases


(Homo sapiens (Human))
BDBM50064176
PNG
(CHEMBL27673 | CHEMBL500996 | METHOCTRAMINE | N,N''...)
Show SMILES COc1ccccc1CNCCCCCCNCCCCCCCCNCCCCCCNCc1ccccc1OC
Show InChI InChI=1S/C36H62N4O2/c1-41-35-23-13-11-21-33(35)31-39-29-19-9-7-17-27-37-25-15-5-3-4-6-16-26-38-28-18-8-10-20-30-40-32-34-22-12-14-24-36(34)42-2/h11-14,21-24,37-40H,3-10,15-20,25-32H2,1-2H3
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n/an/a 977n/an/an/an/an/an/a



University of Bologna

Curated by ChEMBL


Assay Description
Inhibition of Butyrylcholinesterase (BChE) of human erythrocytes [-log IC50 (uM)]


J Med Chem 41: 4186-9 (1998)

Checked by Author
Article DOI: 10.1021/jm9810452
BindingDB Entry DOI: 10.7270/Q2HH6KRM
More data for this
Ligand-Target Pair
Cholinesterases


(Homo sapiens (Human))
BDBM50422272
PNG
(CHEMBL302179)
Show SMILES COc1ccccc1CNCCCCCCNCCCCCCNCCCCCCNCc1ccccc1OC
Show InChI InChI=1S/C34H58N4O2/c1-39-33-21-11-9-19-31(33)29-37-27-17-7-5-15-25-35-23-13-3-4-14-24-36-26-16-6-8-18-28-38-30-32-20-10-12-22-34(32)40-2/h9-12,19-22,35-38H,3-8,13-18,23-30H2,1-2H3
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n/an/a 1.38E+3n/an/an/an/an/an/a



University of Bologna

Curated by ChEMBL


Assay Description
Inhibition of Butyrylcholinesterase (BChE) of human erythrocytes [-log IC50 (uM)]


J Med Chem 41: 4186-9 (1998)

Checked by Author
Article DOI: 10.1021/jm9810452
BindingDB Entry DOI: 10.7270/Q2HH6KRM
More data for this
Ligand-Target Pair
Cholinesterases


(Homo sapiens (Human))
BDBM50422273
PNG
(CHEMBL134488)
Show SMILES COc1ccccc1CNCCCCCC(=O)NCCCCCCCCNC(=O)CCCCCNCc1ccccc1OC
Show InChI InChI=1S/C36H58N4O4/c1-43-33-21-13-11-19-31(33)29-37-25-15-7-9-23-35(41)39-27-17-5-3-4-6-18-28-40-36(42)24-10-8-16-26-38-30-32-20-12-14-22-34(32)44-2/h11-14,19-22,37-38H,3-10,15-18,23-30H2,1-2H3,(H,39,41)(H,40,42)
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n/an/a 1.86E+3n/an/an/an/an/an/a



University of Bologna

Curated by ChEMBL


Assay Description
Inhibition of acetylcholinesterase (AChE) of human erythrocytes


J Med Chem 41: 4186-9 (1998)

Checked by Author
Article DOI: 10.1021/jm9810452
BindingDB Entry DOI: 10.7270/Q2HH6KRM
More data for this
Ligand-Target Pair
Cholinesterases


(Homo sapiens (Human))
BDBM50422270
PNG
(CHEMBL422977)
Show SMILES COc1ccccc1CNCCCCCCNCCCCCCCNCCCCCCNCc1ccccc1OC
Show InChI InChI=1S/C35H60N4O2/c1-40-34-22-12-10-20-32(34)30-38-28-18-8-6-16-26-36-24-14-4-3-5-15-25-37-27-17-7-9-19-29-39-31-33-21-11-13-23-35(33)41-2/h10-13,20-23,36-39H,3-9,14-19,24-31H2,1-2H3
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n/an/a 3.72E+3n/an/an/an/an/an/a



University of Bologna

Curated by ChEMBL


Assay Description
Inhibition of Butyrylcholinesterase (BChE) of human erythrocytes [-log IC50 (uM)]


J Med Chem 41: 4186-9 (1998)

Checked by Author
Article DOI: 10.1021/jm9810452
BindingDB Entry DOI: 10.7270/Q2HH6KRM
More data for this
Ligand-Target Pair
Cholinesterases


(Homo sapiens (Human))
BDBM50422270
PNG
(CHEMBL422977)
Show SMILES COc1ccccc1CNCCCCCCNCCCCCCCNCCCCCCNCc1ccccc1OC
Show InChI InChI=1S/C35H60N4O2/c1-40-34-22-12-10-20-32(34)30-38-28-18-8-6-16-26-36-24-14-4-3-5-15-25-37-27-17-7-9-19-29-39-31-33-21-11-13-23-35(33)41-2/h10-13,20-23,36-39H,3-9,14-19,24-31H2,1-2H3
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n/an/a 4.47E+3n/an/an/an/an/an/a



University of Bologna

Curated by ChEMBL


Assay Description
Inhibition of acetylcholinesterase (AChE) of human erythrocytes


J Med Chem 41: 4186-9 (1998)

Checked by Author
Article DOI: 10.1021/jm9810452
BindingDB Entry DOI: 10.7270/Q2HH6KRM
More data for this
Ligand-Target Pair
Cholinesterases


(Homo sapiens (Human))
BDBM50064176
PNG
(CHEMBL27673 | CHEMBL500996 | METHOCTRAMINE | N,N''...)
Show SMILES COc1ccccc1CNCCCCCCNCCCCCCCCNCCCCCCNCc1ccccc1OC
Show InChI InChI=1S/C36H62N4O2/c1-41-35-23-13-11-21-33(35)31-39-29-19-9-7-17-27-37-25-15-5-3-4-6-16-26-38-28-18-8-10-20-30-40-32-34-22-12-14-24-36(34)42-2/h11-14,21-24,37-40H,3-10,15-20,25-32H2,1-2H3
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n/an/a 5.37E+3n/an/an/an/an/an/a



University of Bologna

Curated by ChEMBL


Assay Description
Inhibition of acetylcholinesterase (AChE) of human erythrocytes


J Med Chem 41: 4186-9 (1998)

Checked by Author
Article DOI: 10.1021/jm9810452
BindingDB Entry DOI: 10.7270/Q2HH6KRM
More data for this
Ligand-Target Pair
Cholinesterases


(Homo sapiens (Human))
BDBM50422269
PNG
(CHEMBL132377)
Show SMILES COc1ccccc1CNCCCCCC(=O)N(C)CCCCCCCCN(C)C(=O)CCCCCNCc1ccccc1OC
Show InChI InChI=1S/C38H62N4O4/c1-41(37(43)25-11-9-17-27-39-31-33-21-13-15-23-35(33)45-3)29-19-7-5-6-8-20-30-42(2)38(44)26-12-10-18-28-40-32-34-22-14-16-24-36(34)46-4/h13-16,21-24,39-40H,5-12,17-20,25-32H2,1-4H3
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n/an/a 6.03E+3n/an/an/an/an/an/a



University of Bologna

Curated by ChEMBL


Assay Description
Inhibition of Butyrylcholinesterase (BChE) of human erythrocytes [-log IC50 (uM)]


J Med Chem 41: 4186-9 (1998)

Checked by Author
Article DOI: 10.1021/jm9810452
BindingDB Entry DOI: 10.7270/Q2HH6KRM
More data for this
Ligand-Target Pair
Cholinesterases


(Homo sapiens (Human))
BDBM50020168
PNG
(1N-(2-methoxybenzyl)-6N-(2-{2-[6-(2-methoxybenzyla...)
Show SMILES COc1ccccc1CNCCCCCCNCCSSCCNCCCCCCNCc1ccccc1OC
Show InChI InChI=1S/C32H54N4O2S2/c1-37-31-17-9-7-15-29(31)27-35-21-13-5-3-11-19-33-23-25-39-40-26-24-34-20-12-4-6-14-22-36-28-30-16-8-10-18-32(30)38-2/h7-10,15-18,33-36H,3-6,11-14,19-28H2,1-2H3
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n/an/a 6.17E+3n/an/an/an/an/an/a



University of Bologna

Curated by ChEMBL


Assay Description
Inhibition of Butyrylcholinesterase (BChE) of human erythrocytes [-log IC50 (uM)]


J Med Chem 41: 4186-9 (1998)

Checked by Author
Article DOI: 10.1021/jm9810452
BindingDB Entry DOI: 10.7270/Q2HH6KRM
More data for this
Ligand-Target Pair
Cholinesterases


(Homo sapiens (Human))
BDBM50422272
PNG
(CHEMBL302179)
Show SMILES COc1ccccc1CNCCCCCCNCCCCCCNCCCCCCNCc1ccccc1OC
Show InChI InChI=1S/C34H58N4O2/c1-39-33-21-11-9-19-31(33)29-37-27-17-7-5-15-25-35-23-13-3-4-14-24-36-26-16-6-8-18-28-38-30-32-20-10-12-22-34(32)40-2/h9-12,19-22,35-38H,3-8,13-18,23-30H2,1-2H3
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n/an/a 6.46E+3n/an/an/an/an/an/a



University of Bologna

Curated by ChEMBL


Assay Description
Inhibition of acetylcholinesterase (AChE) of human erythrocytes


J Med Chem 41: 4186-9 (1998)

Checked by Author
Article DOI: 10.1021/jm9810452
BindingDB Entry DOI: 10.7270/Q2HH6KRM
More data for this
Ligand-Target Pair
Cholinesterases


(Homo sapiens (Human))
BDBM50020168
PNG
(1N-(2-methoxybenzyl)-6N-(2-{2-[6-(2-methoxybenzyla...)
Show SMILES COc1ccccc1CNCCCCCCNCCSSCCNCCCCCCNCc1ccccc1OC
Show InChI InChI=1S/C32H54N4O2S2/c1-37-31-17-9-7-15-29(31)27-35-21-13-5-3-11-19-33-23-25-39-40-26-24-34-20-12-4-6-14-22-36-28-30-16-8-10-18-32(30)38-2/h7-10,15-18,33-36H,3-6,11-14,19-28H2,1-2H3
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Article
PubMed
n/an/a 7.24E+3n/an/an/an/an/an/a



University of Bologna

Curated by ChEMBL


Assay Description
Inhibition of acetylcholinesterase (AChE) of human erythrocytes


J Med Chem 41: 4186-9 (1998)

Checked by Author
Article DOI: 10.1021/jm9810452
BindingDB Entry DOI: 10.7270/Q2HH6KRM
More data for this
Ligand-Target Pair
Cholinesterases


(Homo sapiens (Human))
BDBM50422271
PNG
(CHEMBL134382)
Show SMILES COc1ccccc1CNCCCCCCNCCCCCNCCCCCCNCc1ccccc1OC
Show InChI InChI=1S/C33H56N4O2/c1-38-32-20-10-8-18-30(32)28-36-26-14-5-3-12-22-34-24-16-7-17-25-35-23-13-4-6-15-27-37-29-31-19-9-11-21-33(31)39-2/h8-11,18-21,34-37H,3-7,12-17,22-29H2,1-2H3
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PubMed
n/an/a 7.24E+3n/an/an/an/an/an/a



University of Bologna

Curated by ChEMBL


Assay Description
Inhibition of acetylcholinesterase (AChE) of human erythrocytes


J Med Chem 41: 4186-9 (1998)

Checked by Author
Article DOI: 10.1021/jm9810452
BindingDB Entry DOI: 10.7270/Q2HH6KRM
More data for this
Ligand-Target Pair
Cholinesterases


(Homo sapiens (Human))
BDBM50422271
PNG
(CHEMBL134382)
Show SMILES COc1ccccc1CNCCCCCCNCCCCCNCCCCCCNCc1ccccc1OC
Show InChI InChI=1S/C33H56N4O2/c1-38-32-20-10-8-18-30(32)28-36-26-14-5-3-12-22-34-24-16-7-17-25-35-23-13-4-6-15-27-37-29-31-19-9-11-21-33(31)39-2/h8-11,18-21,34-37H,3-7,12-17,22-29H2,1-2H3
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n/an/a 8.71E+3n/an/an/an/an/an/a



University of Bologna

Curated by ChEMBL


Assay Description
Inhibition of Butyrylcholinesterase (BChE) of human erythrocytes [-log IC50 (uM)]


J Med Chem 41: 4186-9 (1998)

Checked by Author
Article DOI: 10.1021/jm9810452
BindingDB Entry DOI: 10.7270/Q2HH6KRM
More data for this
Ligand-Target Pair
Cholinesterases


(Homo sapiens (Human))
BDBM50422273
PNG
(CHEMBL134488)
Show SMILES COc1ccccc1CNCCCCCC(=O)NCCCCCCCCNC(=O)CCCCCNCc1ccccc1OC
Show InChI InChI=1S/C36H58N4O4/c1-43-33-21-13-11-19-31(33)29-37-25-15-7-9-23-35(41)39-27-17-5-3-4-6-18-28-40-36(42)24-10-8-16-26-38-30-32-20-12-14-22-34(32)44-2/h11-14,19-22,37-38H,3-10,15-18,23-30H2,1-2H3,(H,39,41)(H,40,42)
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n/an/a 1.15E+4n/an/an/an/an/an/a



University of Bologna

Curated by ChEMBL


Assay Description
Inhibition of Butyrylcholinesterase (BChE) of human erythrocytes [-log IC50 (uM)]


J Med Chem 41: 4186-9 (1998)

Checked by Author
Article DOI: 10.1021/jm9810452
BindingDB Entry DOI: 10.7270/Q2HH6KRM
More data for this
Ligand-Target Pair
Cholinesterases


(Homo sapiens (Human))
BDBM50067482
PNG
(6-[(2-Methoxy-benzyl)-methyl-amino]-hexanoic acid ...)
Show SMILES COc1ccccc1CN(C)CCCCCC(=O)N(C)CCCCCCCCN(C)C(=O)CCCCCN(C)Cc1ccccc1OC
Show InChI InChI=1S/C40H66N4O4/c1-41(33-35-23-15-17-25-37(35)47-5)29-19-11-13-27-39(45)43(3)31-21-9-7-8-10-22-32-44(4)40(46)28-14-12-20-30-42(2)34-36-24-16-18-26-38(36)48-6/h15-18,23-26H,7-14,19-22,27-34H2,1-6H3
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n/an/a 1.17E+4n/an/an/an/an/an/a



University of Bologna

Curated by ChEMBL


Assay Description
Inhibition of Butyrylcholinesterase (BChE) of human erythrocytes [-log IC50 (uM)]


J Med Chem 41: 4186-9 (1998)

Checked by Author
Article DOI: 10.1021/jm9810452
BindingDB Entry DOI: 10.7270/Q2HH6KRM
More data for this
Ligand-Target Pair
Cholinesterases


(Homo sapiens (Human))
BDBM50455151
PNG
(CHEMBL132133)
Show SMILES NCCCCCCNCCSSCCNCCCCCCN
Show InChI InChI=1S/C16H38N4S2/c17-9-5-1-3-7-11-19-13-15-21-22-16-14-20-12-8-4-2-6-10-18/h19-20H,1-18H2
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n/an/a 5.01E+5n/an/an/an/an/an/a



University of Bologna

Curated by ChEMBL


Assay Description
Inhibition of acetylcholinesterase (AChE) of human erythrocytes


J Med Chem 41: 4186-9 (1998)

Checked by Author
Article DOI: 10.1021/jm9810452
BindingDB Entry DOI: 10.7270/Q2HH6KRM
More data for this
Ligand-Target Pair
Cholinesterases


(Homo sapiens (Human))
BDBM50455151
PNG
(CHEMBL132133)
Show SMILES NCCCCCCNCCSSCCNCCCCCCN
Show InChI InChI=1S/C16H38N4S2/c17-9-5-1-3-7-11-19-13-15-21-22-16-14-20-12-8-4-2-6-10-18/h19-20H,1-18H2
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n/an/a 6.46E+5n/an/an/an/an/an/a



University of Bologna

Curated by ChEMBL


Assay Description
Inhibition of Butyrylcholinesterase (BChE) of human erythrocytes [-log IC50 (uM)]


J Med Chem 41: 4186-9 (1998)

Checked by Author
Article DOI: 10.1021/jm9810452
BindingDB Entry DOI: 10.7270/Q2HH6KRM
More data for this
Ligand-Target Pair
* indicates data uncertainty>20%