Reaction Details Report a problem with these data
Target
Eukaryotic initiation factor 4A-II
Ligand
BDBM65493
Substrate
n/a
Meas. Tech.
ATPase enzyme assay
IC50
>1.00e+5±n/a nM
Citation
Iwatani-Yoshihara, M; Ito, M; Ishibashi, Y; Oki, H; Tanaka, T; Morishita, D; Ito, T; Kimura, H; Imaeda, Y; Aparicio, S; Nakanishi, A; Kawamoto, T Discovery and Characterization of a Eukaryotic Initiation Factor 4A-3-Selective Inhibitor That Suppresses Nonsense-Mediated mRNA Decay. ACS Chem Biol 12:1760-1768 (2017) [PubMed] Article
More Info.:
Target
Name:
Eukaryotic initiation factor 4A-II
Synonyms:
ATP-dependent RNA helicase eIF4A-2 | DDX2B | EIF4A2 | EIF4F | IF4A2_HUMAN | eIF-4A-II | eIF4A-II
Type:
Protein
Mol. Mass.:
46394.69
Organism:
Homo sapiens (Human)
Description:
Q14240
Residue:
407
Sequence:
MSGGSADYNREHGGPEGMDPDGVIESNWNEIVDNFDDMNLKESLLRGIYAYGFEKPSAIQQRAIIPCIKGYDVIAQAQSGTGKTATFAISILQQLEIEFKETQALVLAPTRELAQQIQKVILALGDYMGATCHACIGGTNVRNEMQKLQAEAPHIVVGTPGRVFDMLNRRYLSPKWIKMFVLDEADEMLSRGFKDQIYEIFQKLNTSIQVVLLSATMPTDVLEVTKKFMRDPIRILVKKEELTLEGIKQFYINVEREEWKLDTLCDLYETLTITQAVIFLNTRRKVDWLTEKMHARDFTVSALHGDMDQKERDVIMREFRSGSSRVLITTDLLARGIDVQQVSLVINYDLPTNRENYIHRIGRGGRFGRKGVAINFVTEEDKRILRDIETFYNTTVEEMPMNVADLI