Reaction Details Report a problem with these data
Target
N-formyl peptide receptor 2
Ligand
BDBM37721
Substrate
n/a
Meas. Tech.
Dose Response Assay for Formylpeptide Receptor-Like-1 (FPRL1) Ligands and Dose Response Counter-Screen Assay for Formylpeptide Receptor (FPR) Ligands
Ki
11000±n/a nM
Comments
Extracted from aid = 520 and tid = 2
Citation
 PubChem, PC Dose Response Assay for Formylpeptide Receptor-Like-1 (FPRL1) Ligands and Dose Response Counter-Screen Assay for Formylpeptide Receptor (FPR) Ligands PubChem Bioassay (2007)[AID] 
Target
Name:
N-formyl peptide receptor 2
Synonyms:
ALXR, FPRL1, FPR2 | FMLP-related receptor I FMLP-R-I | FPR2 | FPR2_HUMAN | FPRH1 | FPRL1 | Formyl Peptide Receptor-Like 1 | HM63 | LXA4 receptor | LXA4R | Lipoxin A4 receptor | Lipoxin A4 receptor (LXA4) | RFP | hFPRL
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
38968.35
Organism:
Homo sapiens (Human)
Description:
P25090
Residue:
351
Sequence:
METNFSTPLNEYEEVSYESAGYTVLRILPLVVLGVTFVLGVLGNGLVIWVAGFRMTRTVTTICYLNLALADFSFTATLPFLIVSMAMGEKWPFGWFLCKLIHIVVDINLFGSVFLIGFIALDRCICVLHPVWAQNHRTVSLAMKVIVGPWILALVLTLPVFLFLTTVTIPNGDTYCTFNFASWGGTPEERLKVAITMLTARGIIRFVIGFSLPMSIVAICYGLIAAKIHKKGMIKSSRPLRVLTAVVASFFICWFPFQLVALLGTVWLKEMLFYGKYKIIDILVNPTSSLAFFNSCLNPMLYVFVGQDFRERLIHSLPTSLERALSEDSAPTNDTAANSASPPAETELQAM
  
Inhibitor
Name:
BDBM37721
Synonyms:
2-(3-chlorophenyl)-4-N-methyltriazole-4,5-diamine | 2-(3-chlorophenyl)-N-methyl-2H-1,2,3-triazole-4,5-diamine | 2-(3-chlorophenyl)-N4-methyl-1,2,3-triazole-4,5-diamine | 2-(3-chlorophenyl)-N4-methyltriazole-4,5-diamine | MLS000091276 | SMR000025838 | [5-amino-2-(3-chlorophenyl)triazol-4-yl]-methyl-amine | cid_3240793
Type:
Small organic molecule
Emp. Form.:
C9H10ClN5
Mol. Mass.:
223.662
SMILES:
CNc1nn(nc1N)-c1cccc(Cl)c1
Structure:
Search PDB for entries with ligand similarity: