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Target
Matrix metalloproteinase-14 [1-36]
Ligand
BDBM39020
Substrate
n/a
Meas. Tech.
Luminescent HTS for small molecule inhibitors of MT1-MMP transcription
EC50
820±n/a nM
Citation
 PubChem, PC Luminescent HTS for small molecule inhibitors of MT1-MMP transcription PubChem Bioassay (2008)[AID] 
Target
Name:
Matrix metalloproteinase-14 [1-36]
Synonyms:
MMP14 | MMP14_PONAB | matrix metalloproteinase 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
3658.23
Organism:
Homo sapiens (Human)
Description:
gi_6690534
Residue:
36
Sequence:
MSPAPRPSRCLLLPLLTLGTALASLGSAQSSSFSPE
  
Inhibitor
Name:
BDBM39020
Synonyms:
3-[(4,5-dimethyl-2-furoyl)amino]benzoic acid | 3-[(4,5-dimethylfuran-2-carbonyl)amino]benzoic acid | 3-[(4,5-dimethylfuran-2-yl)carbonylamino]benzoic acid | 3-[[(4,5-dimethyl-2-furanyl)-oxomethyl]amino]benzoic acid | MLS000062053 | SMR000070049 | cid_781047
Type:
Small organic molecule
Emp. Form.:
C14H13NO4
Mol. Mass.:
259.2573
SMILES:
Cc1cc(oc1C)C(=O)Nc1cccc(c1)C(O)=O
Structure:
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