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Target
Matrix metalloproteinase-14 [1-36]
Ligand
BDBM48217
Substrate
n/a
Meas. Tech.
Luminescent HTS for small molecule inhibitors of MT1-MMP transcription
EC50
280±n/a nM
Citation
 PubChem, PC Luminescent HTS for small molecule inhibitors of MT1-MMP transcription PubChem Bioassay (2008)[AID] 
Target
Name:
Matrix metalloproteinase-14 [1-36]
Synonyms:
MMP14 | MMP14_PONAB | matrix metalloproteinase 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
3658.23
Organism:
Homo sapiens (Human)
Description:
gi_6690534
Residue:
36
Sequence:
MSPAPRPSRCLLLPLLTLGTALASLGSAQSSSFSPE
  
Inhibitor
Name:
BDBM48217
Synonyms:
1-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-4-phenyl-butan-1-one | 1-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-phenyl-1-butanone | 1-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-phenyl-butan-1-one | 1-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-phenylbutan-1-one | MLS000525661 | SMR000116135 | cid_3129671
Type:
Small organic molecule
Emp. Form.:
C18H18O3
Mol. Mass.:
282.3337
SMILES:
O=C(CCCc1ccccc1)c1ccc2OCCOc2c1
Structure:
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