Target
Matrix metalloproteinase-14 [1-36]
Ligand
BDBM48256
Substrate
n/a
Meas. Tech.
Luminescent HTS for small molecule inhibitors of MT1-MMP transcription
EC50
660±n/a nM
Citation
 PubChem, PC Luminescent HTS for small molecule inhibitors of MT1-MMP transcription PubChem Bioassay (2008)[AID] 
Target
Name:
Matrix metalloproteinase-14 [1-36]
Synonyms:
MMP14 | MMP14_PONAB | matrix metalloproteinase 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
3658.23
Organism:
Homo sapiens (Human)
Description:
gi_6690534
Residue:
36
Sequence:
MSPAPRPSRCLLLPLLTLGTALASLGSAQSSSFSPE
  
Inhibitor
Name:
BDBM48256
Synonyms:
3-(p-toluoylamino)benzoic acid | 3-[(4-methylbenzoyl)amino]benzoic acid | 3-[(4-methylphenyl)carbonylamino]benzoic acid | 3-[[(4-methylphenyl)-oxomethyl]amino]benzoic acid | MLS000530214 | SMR000135191 | cid_735216
Type:
Small organic molecule
Emp. Form.:
C15H13NO3
Mol. Mass.:
255.2686
SMILES:
Cc1ccc(cc1)C(=O)Nc1cccc(c1)C(O)=O
Structure:
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