Reaction Details Report a problem with these data
Target
Neuropeptide Y receptor type 1
Ligand
BDBM58038
Substrate
n/a
Meas. Tech.
Fluorescence-based dose response cell-based high-throughput screening assay for potentiators or agonists of NPY-Y1.
EC50
10072±n/a nM
Citation
 PubChem, PC Fluorescence-based dose response cell-based high-throughput screening assay for potentiators or agonists of NPY-Y1. PubChem Bioassay (2009)[AID] 
Target
Name:
Neuropeptide Y receptor type 1
Synonyms:
NPY-Y1 | NPY1-R | NPY1R | NPY1R_HUMAN | NPYR | NPYY1 | neuropeptide Y receptor Y1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
44399.07
Organism:
Homo sapiens (Human)
Description:
NPY-Y1 NPY1R HUMAN::P25929
Residue:
384
Sequence:
MNSTLFSQVENHSVHSNFSEKNAQLLAFENDDCHLPLAMIFTLALAYGAVIILGVSGNLALIIIILKQKEMRNVTNILIVNLSFSDLLVAIMCLPFTFVYTLMDHWVFGEAMCKLNPFVQCVSITVSIFSLVLIAVERHQLIINPRGWRPNNRHAYVGIAVIWVLAVASSLPFLIYQVMTDEPFQNVTLDAYKDKYVCFDQFPSDSHRLSYTTLLLVLQYFGPLCFIFICYFKIYIRLKRRNNMMDKMRDNKYRSSETKRINIMLLSIVVAFAVCWLPLTIFNTVFDWNHQIIATCNHNLLFLLCHLTAMISTCVNPIFYGFLNKNFQRDLQFFFNFCDFRSRDDDYETIAMSTMHTDVSKTSLKQASPVAFKKINNNDDNEKI
  
Inhibitor
Name:
BDBM58038
Synonyms:
2-(3-Bromo-phenyl)-3-(4-chloro-phenyl)-1H-imidazo[4,5-b]quinoxaline | 2-(3-bromophenyl)-3-(4-chlorophenyl)-1H-imidazo[4,5-b]quinoxalin-3-ium | MLS001012274 | SMR000425093 | cid_5604367
Type:
Small organic molecule
Emp. Form.:
C21H13BrClN4
Mol. Mass.:
436.711
SMILES:
Clc1ccc(cc1)-[n+]1c([nH]c2nc3ccccc3nc12)-c1cccc(Br)c1
Structure:
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