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Target
Trans-activator protein BZLF1
Ligand
BDBM64848
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of PP1: fluorescence-based biochemical high throughput dose response assay to identify inhibitors of Protein Phosphatase 5 (PP5)
IC50
37949±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of PP1: fluorescence-based biochemical high throughput dose response assay to identify inhibitors of Protein Phosphatase 5 (PP5) PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM64848
Synonyms:
1,3-benzodioxol-5-yl-[7-methyl-2-(2-pyridyl)imidazo[1,2-a]pyridin-3-yl]amine | MLS000580787 | N-(1,3-benzodioxol-5-yl)-7-methyl-2-(2-pyridinyl)-3-imidazo[1,2-a]pyridinamine | N-(1,3-benzodioxol-5-yl)-7-methyl-2-pyridin-2-yl-imidazo[1,2-a]pyridin-3-amine | N-(1,3-benzodioxol-5-yl)-7-methyl-2-pyridin-2-ylimidazo[1,2-a]pyridin-3-amine | N-1,3-benzodioxol-5-yl-7-methyl-2-pyridin-2-ylimidazo[1,2-a]pyridin-3-amine | SMR000206173 | cid_12004827
Type:
Small organic molecule
Emp. Form.:
C20H16N4O2
Mol. Mass.:
344.3666
SMILES:
Cc1ccn2c(Nc3ccc4OCOc4c3)c(nc2c1)-c1ccccn1
Structure:
Search PDB for entries with ligand similarity: