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Target
Trans-activator protein BZLF1
Ligand
BDBM64859
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of PP1: fluorescence-based biochemical high throughput dose response assay to identify inhibitors of Protein Phosphatase 5 (PP5)
IC50
62230±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of PP1: fluorescence-based biochemical high throughput dose response assay to identify inhibitors of Protein Phosphatase 5 (PP5) PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM64859
Synonyms:
5-[(2-chloranyl-6-fluoranyl-phenyl)methyl]-2-pyridin-2-yl-pyrimidine-4,6-diamine | 5-[(2-chloro-6-fluorophenyl)methyl]-2-(2-pyridinyl)pyrimidine-4,6-diamine | 5-[(2-chloro-6-fluorophenyl)methyl]-2-pyridin-2-ylpyrimidine-4,6-diamine | 6-amino-5-(2-chloro-6-fluorobenzyl)-2-(2-pyridinyl)-4-pyrimidinylamine | MLS000691909 | SMR000333932 | [6-amino-5-(2-chloro-6-fluoro-benzyl)-2-(2-pyridyl)pyrimidin-4-yl]amine | cid_4667754
Type:
Small organic molecule
Emp. Form.:
C16H13ClFN5
Mol. Mass.:
329.759
SMILES:
Nc1nc(nc(N)c1Cc1c(F)cccc1Cl)-c1ccccn1
Structure:
Search PDB for entries with ligand similarity: