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Target
Trans-activator protein BZLF1
Ligand
BDBM64861
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of PP1: fluorescence-based biochemical high throughput dose response assay to identify inhibitors of Protein Phosphatase 5 (PP5)
IC50
47473±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of PP1: fluorescence-based biochemical high throughput dose response assay to identify inhibitors of Protein Phosphatase 5 (PP5) PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM64861
Synonyms:
5-(2,4-dichlorobenzyl)-2-(2-pyridinyl)-4,6-pyrimidinediamine | 5-[(2,4-dichlorophenyl)methyl]-2-(2-pyridinyl)pyrimidine-4,6-diamine | 5-[(2,4-dichlorophenyl)methyl]-2-pyridin-2-yl-pyrimidine-4,6-diamine | 5-[(2,4-dichlorophenyl)methyl]-2-pyridin-2-ylpyrimidine-4,6-diamine | MLS000691892 | SMR000333929 | [6-amino-5-(2,4-dichlorobenzyl)-2-(2-pyridyl)pyrimidin-4-yl]amine | cid_3379829
Type:
Small organic molecule
Emp. Form.:
C16H13Cl2N5
Mol. Mass.:
346.214
SMILES:
Nc1nc(nc(N)c1Cc1ccc(Cl)cc1Cl)-c1ccccn1
Structure:
Search PDB for entries with ligand similarity: