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TargetAryl hydrocarbon receptor
LigandBDBM51199
Substrate/Competitorn/a
Meas. Tech.Luminescence-based cell-based high throughput dose response assay for activators of the Aryl Hydrocarbon Receptor (AHR)
EC50 4820±n/a nM
Citation PubChem, PC Luminescence-based cell-based high throughput dose response assay for activators of the Aryl Hydrocarbon Receptor (AHR) PubChem Bioassay(2010)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Aryl hydrocarbon receptor
Name:Aryl hydrocarbon receptor
Synonyms:AhR | Class E basic helix-loop-helix protein 76 | aryl hydrocarbon receptor precursor | bHLHe76
Type:PROTEIN
Mol. Mass.:96143.77
Organism:Homo sapiens (Human)
Description:ChEMBL_1503828
Residue:848
Sequence:
MNSSSANITYASRKRRKPVQKTVKPIPAEGIKSNPSKRHRDRLNTELDRLASLLPFPQDV
INKLDKLSVLRLSVSYLRAKSFFDVALKSSPTERNGGQDNCRAANFREGLNLQEGEFLLQ
ALNGFVLVVTTDALVFYASSTIQDYLGFQQSDVIHQSVYELIHTEDRAEFQRQLHWALNP
SQCTESGQGIEEATGLPQTVVCYNPDQIPPENSPLMERCFICRLRCLLDNSSGFLAMNFQ
GKLKYLHGQKKKGKDGSILPPQLALFAIATPLQPPSILEIRTKNFIFRTKHKLDFTPIGC
DAKGRIVLGYTEAELCTRGSGYQFIHAADMLYCAESHIRMIKTGESGMIVFRLLTKNNRW
TWVQSNARLLYKNGRPDYIIVTQRPLTDEEGTEHLRKRNTKLPFMFTTGEAVLYEATNPF
PAIMDPLPLRTKNGTSGKDSATTSTLSKDSLNPSSLLAAMMQQDESIYLYPASSTSSTAP
FENNFFNESMNECRNWQDNTAPMGNDTILKHEQIDQPQDVNSFAGGHPGLFQDSKNSDLY
SIMKNLGIDFEDIRHMQNEKFFRNDFSGEVDFRDIDLTDEILTYVQDSLSKSPFIPSDYQ
QQQSLALNSSCMVQEHLHLEQQQQHHQKQVVVEPQQQLCQKMKHMQVNGMFENWNSNQFV
PFNCPQQDPQQYNVFTDLHGISQEFPYKSEMDSMPYTQNFISCNQPVLPQHSKCTELDYP
MGSFEPSPYPTTSSLEDFVTCLQLPENQKHGLNPQSAIITPQTCYAGAVSMYQCQPEPQH
THVGQMQYNPVLPGQQAFLNKFQNGVLNETYPAELNNINNTQTTTHLQPLHHPSEARPFP
DLTSSGFL
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  Blast E-value cutoff:
BDBM51199
NameBDBM51199
Synonyms:2-(6-nitro-2-phenyl-benzimidazol-1-yl)oxyacetic acid | 2-(6-nitro-2-phenyl-benzimidazol-1-yl)oxyethanoic acid | 2-(6-nitro-2-phenylbenzimidazol-1-yl)oxyacetic acid | 2-[(6-nitro-2-phenyl-1-benzimidazolyl)oxy]acetic acid | 2-[(6-nitro-2-phenyl-1H-1,3-benzimidazol-1-yl)oxy]acetic acid | MLS000755385 | SMR000337780 | cid_2766807
TypeSmall organic molecule
Emp. Form.C15H11N3O5
Mol. Mass.313.2649
SMILESOC(=O)COn1c(nc2ccc(cc12)[N+]([O-])=O)-c1ccccc1
Structure
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n/a