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Targetubiquitin-conjugating enzyme E2 N
LigandBDBM79379
Substrate/Competitorn/a
Meas. Tech.Dose Response confirmation of uHTS for the identification of UBC13 Polyubiquitin Inhibitors via a TR-FRET Assay
IC50>20000±0 nM
Citation PubChem, PC Dose Response confirmation of uHTS for the identification of UBC13 Polyubiquitin Inhibitors via a TR-FRET Assay PubChem Bioassay(2011)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
ubiquitin-conjugating enzyme E2 N
Name:Ubiquitin-conjugating enzyme E2 N
Synonyms:n/a
Type:PROTEIN
Mol. Mass.:17137.61
Organism:Homo sapiens (Human)
Description:EBI_101440
Residue:152
Sequence:
MAGLPRRIIKETQRLLAEPVPGIKAEPDESNARYFHVVIAGPQDSPFEGGTFKLELFLPE
EYPMAAPKVRFMTKIYHPNVDKLGRICLDILKDKWSPALQIRTVLLSIQALLSAPNPDDP
LANDVAEQWKTNEAQAIETARAWTRLYAMNNI
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM79379
NameBDBM79379
Synonyms:3-[[(6-chloranylpyridin-3-yl)carbonylamino]carbamoyl]-N-(2-methoxyphenyl)benzenesulfonamide | 3-[[(6-chloronicotinoyl)amino]carbamoyl]-N-(2-methoxyphenyl)benzenesulfonamide | 3-[[(6-chloropyridine-3-carbonyl)amino]carbamoyl]-N-(2-methoxyphenyl)benzenesulfonamide | 3-[[[(6-chloro-3-pyridinyl)-oxomethyl]hydrazo]-oxomethyl]-N-(2-methoxyphenyl)benzenesulfonamide | MLS002248406 | SMR001315877 | cid_2081452
TypeSmall organic molecule
Emp. Form.C20H17ClN4O5S
Mol. Mass.460.891
SMILESCOc1ccccc1NS(=O)(=O)c1cccc(c1)C(=O)NNC(=O)c1ccc(Cl)nc1
Structure
Search PDB for entries with ligand similarity:Similarity to this molecule at least:
n/a