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Target
Beta-2 adrenergic receptor
Ligand
BDBM50292375
Substrate
n/a
Ki
>10000±n/a nM
Comments
PDSP_1789
Citation
 Bylund, DB; Snyder, SH Beta adrenergic receptor binding in membrane preparations from mammalian brain. Mol Pharmacol 12:568-80 (1976) [PubMed] 
Target
Name:
Beta-2 adrenergic receptor
Synonyms:
ADRB2 | ADRB2R | ADRB2_HUMAN | B2AR | Beta-2 adrenoceptor | Beta-2 adrenoreceptor
Type:
n/a
Mol. Mass.:
46461.69
Organism:
Homo sapiens (Human)
Description:
P07550
Residue:
413
Sequence:
MGQPGNGSAFLLAPNGSHAPDHDVTQERDEVWVVGMGIVMSLIVLAIVFGNVLVITAIAKFERLQTVTNYFITSLACADLVMGLAVVPFGAAHILMKMWTFGNFWCEFWTSIDVLCVTASIETLCVIAVDRYFAITSPFKYQSLLTKNKARVIILMVWIVSGLTSFLPIQMHWYRATHQEAINCYANETCCDFFTNQAYAIASSIVSFYVPLVIMVFVYSRVFQEAKRQLQKIDKSEGRFHVQNLSQVEQDGRTGHGLRRSSKFCLKEHKALKTLGIIMGTFTLCWLPFFIVNIVHVIQDNLIRKEVYILLNWIGYVNSGFNPLIYCRSPDFRIAFQELLCLRRSSLKAYGNGYSSNGNTGEQSGYHVEQEKENKLLCEDLPGTEDFVGHQGTVPSDNIDSQGRNCSTNDSLL
  
Inhibitor
Name:
BDBM50292375
Synonyms:
(-)-4-hydroxy-alpha-[(methylamino)methyl]benzenemethanol | (-)-Oxedrine | (-)-Sympatol | (-)-Synephrine | (-)-p-hydroxy-alpha-[(methylamino)methyl]benzyl alcohol | 4-[(1R)-1-hydroxy-2-(methylamino)ethyl]phenol | CHEMBL443893 | D(-)-Synephrine | D-synephrine | Synephrine,(+/-)
Type:
Small organic molecule
Emp. Form.:
C9H13NO2
Mol. Mass.:
167.205
SMILES:
CNC[C@H](O)c1ccc(O)cc1 |r|
Structure:
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