Reaction Details Report a problem with these data
Target
Alpha-2C adrenergic receptor
Ligand
BDBM81807
Substrate
n/a
Ki
0.46±n/a nM
Comments
PDSP_332
Citation
 Blaxall, HS; Murphy, TJ; Baker, JC; Ray, C; Bylund, DB Characterization of the alpha-2C adrenergic receptor subtype in the opossum kidney and in the OK cell line. J Pharmacol Exp Ther 259:323-9 (1991) [PubMed] 
Target
Name:
Alpha-2C adrenergic receptor
Synonyms:
ADRA2C | adrenergic Alpha2C
Type:
Enzyme Catalytic Domain
Mol. Mass.:
27257.01
Organism:
OK
Description:
adrenergic Alpha2C ADRA2C OK::G3GWB4
Residue:
230
Sequence:
MAYWYFGQVWCGVYLALDVLFCTSSIVHLCAISLDRYWSVTQAVEYNLKRTPRRVKATIVAVWLISAVISFPPLVSFYRRSDGAAYPQCGLNDETWYILSSCIGSFFAPCLIMGLVYARIYRFFLSRRRRARSSVCRRKVAQAREKRFTFVLAVVMGVFVLCWFPFFFSYSLYGICREACQLPEPLFKFFFWIGYCKSSLNPVIYTVFNQDFRRSFKHILFRRRRRGFRQ
  
Inhibitor
Name:
BDBM81807
Synonyms:
ATIPAMEZOLE | CAS_104054-27-5 | NSC_71310
Type:
Small organic molecule
Emp. Form.:
C14H16N2
Mol. Mass.:
212.2902
SMILES:
CCC1(Cc2ccccc2C1)c1cnc[nH]1
Structure:
Search PDB for entries with ligand similarity: