Reaction Details Report a problem with these data
Target
Alpha-2C adrenergic receptor
Ligand
BDBM81444
Substrate
n/a
Ki
1.6±n/a nM
Comments
PDSP_1955
Citation
Blaxall, HS; Murphy, TJ; Baker, JC; Ray, C; Bylund, DB Characterization of the alpha-2C adrenergic receptor subtype in the opossum kidney and in the OK cell line. J Pharmacol Exp Ther 259:323-9 (1991) [PubMed]
More Info.:
Target
Name:
Alpha-2C adrenergic receptor
Synonyms:
ADA2C_DIDVI | ADRA2C | Alpha-2C adrenergic receptor | adrenergic Alpha2C
Type:
Enzyme Catalytic Domain
Mol. Mass.:
53254.77
Organism:
OPOSSUM
Description:
adrenergic Alpha2C ADRA2C OPOSSUM::P35405
Residue:
469
Sequence:
MDLQLTTNSTDSGDRGGSSNESLQRQPPSQYSPAEVAGLAAVVSFLIVFTIVGNVLVVIAVLTSRALKAPQNLFQVSLASADILVATLVMPFSLANELMNYWYFGKVWCVIYLALDVLFCTSSIVHLCAISLDRYWSVTQAVEYNLKRTPRRIKGIIVTVWLISAVISFPPLISLYRDPEDDLYPQCELNDETWYILSSCIGSFFAPCIIMVLVYVRIYRVAKLRTRTLSEKRTVPEGSSQTENGLSRPPVGAGPSTAAAAAASLRLQAGENGHYHLHHHHHHLHHHHHHHHHQLRKSAELEDIELEESSTSENRRRRRSREEAAARKGSRGFSFSFSSTKGGQSAGAGSRLSRASNRSLEFFSTHRRRKRSSLCRRKVTQAREKRFTFVLAVVMGVFVVCWFPFFFTYSLYGICREACQVPETLFKFFFWIGYCNSSLNPVIYTIFNQDFRRSFKHILFKKKKKTSLQ