Target
Norepinephrine transporter
Ligand
BDBM82219
Substrate
n/a
Ki
18±n/a nM
Comments
PDSP_4195
Citation
 Koe, BKWeissman, AWelch, WMBrowne, RG Sertraline, 1S,4S-N-methyl-4-(3,4-dichlorophenyl)-1,2,3,4-tetrahydro-1-naphthylamine, a new uptake inhibitor with selectivity for serotonin. J Pharmacol Exp Ther 226:686-700 (1983) [PubMed] 
Target
Name:
Norepinephrine transporter
Synonyms:
n/a
Type:
Enzyme Catalytic Domain
Mol. Mass.:
2082.45
Organism:
RAT
Description:
Norepinephrine transporter 0 RAT::Q9JIA2
Residue:
19
Sequence:
MLLARMKPQVQPELGGADQ
  
Inhibitor
Name:
BDBM82219
Synonyms:
CAS_52760-47-1 | CHEMBL38120 | CP-24441 | Tametraline hydrochloride
Type:
Small organic molecule
Emp. Form.:
C17H19N
Mol. Mass.:
237.3395
SMILES:
CN[C@@H]1CC[C@@H](c2ccccc2)c2ccccc12
Structure:
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