Reaction Details Report a problem with these data
Target
Cholecystokinin
Ligand
BDBM82243
Substrate
n/a
Ki
>10000±n/a nM
Comments
PDSP_2678
Citation
 Van Dijk, A; Richards, JG; Trzeciak, A; Gillessen, D; Möhler, H Cholecystokinin receptors: biochemical demonstration and autoradiographical localization in rat brain and pancreas using [3H] cholecystokinin8 as radioligand. J Neurosci 4:1021-33 (1984) [PubMed] 
Target
Name:
Cholecystokinin
Synonyms:
CCKN_RAT | Cck
Type:
Enzyme Catalytic Domain
Mol. Mass.:
12844.29
Organism:
RAT
Description:
Cholecystokinin 0 RAT::P01355
Residue:
115
Sequence:
MKCGVCLCVVMAVLAAGALAQPVVPVEAVDPMEQRAEEAPRRQLRAVLRPDSEPRARLGALLARYIQQVRKAPSGRMSVLKNLQGLDPSHRISDRDYMGWMDFGRRSAEDYEYPS
  
Inhibitor
Name:
BDBM82243
Synonyms:
CCK4 acid
Type:
Small organic molecule
Emp. Form.:
C31H38N6O8
Mol. Mass.:
622.6688
SMILES:
CC(C)CC(NC(=O)C(N)Cc1c[nH]c2ccccc12)C(=O)NC(CC(O)=O)C(=O)NC(Cc1ccccc1)C(=O)NC(O)=O
Structure:
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