Reaction Details Report a problem with these data
Target
Nicotinic acetylcholine receptor
Ligand
BDBM10759
Substrate
n/a
Ki
47.3±n/a nM
Comments
PDSP_229
Citation
 Houghtling, RA; Dávila-García, MI; Kellar, KJ Characterization of (+/-)(-)[3H]epibatidine binding to nicotinic cholinergic receptors in rat and human brain. Mol Pharmacol 48:280-7 (1995) [PubMed] 
Target
Name:
Nicotinic acetylcholine receptor
Synonyms:
Nicotinic acetylcholine receptor | n-AChR
Type:
Enzyme Catalytic Domain
Mol. Mass.:
2478.99
Organism:
RAT
Description:
n-AChR 0 RAT::Q62594
Residue:
23
Sequence:
MTMALLGTLLLLALFGRSQGKNE
  
Inhibitor
Name:
BDBM10759
Synonyms:
2-acetoxyethyl(trimethyl)ammonium;bromide | 2-acetoxyethyl(trimethyl)ammonium;perchlorate | CHEMBL667 | US10667515, Compound ACh | [2-(acetyloxy)ethyl]trimethylazanium | acetylcholine | acetylcholine chloride | cid_6060
Type:
Small Organic Molecule
Emp. Form.:
C7H16NO2
Mol. Mass.:
146.2069
SMILES:
CC(=O)OCC[N+](C)(C)C
Structure:
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