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Target
GABA(A) receptor-associated protein
Ligand
BDBM82387
Substrate
n/a
Ki
7800±n/a nM
Comments
PDSP_48
Citation
Evans, BE; Bock, MG; Rittle, KE; DiPardo, RM; Whitter, WL; Veber, DF; Anderson, PS; Freidinger, RM Design of potent, orally effective, nonpeptidal antagonists of the peptide hormone cholecystokinin. Proc Natl Acad Sci U S A 83:4918-22 (1986) [PubMed] Article
More Info.:
Target
Name:
GABA(A) receptor-associated protein
Synonyms:
GABA A Benzodiazepine | GABA-A receptor subunit alpha 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
13921.89
Organism:
GUINEA PIG
Description:
D7RA28
Residue:
117
Sequence:
MKFVYKEEHPFEKRRSEGEKIRKKYPDRVPVIVEKAPKARIGDLDKKKYLVPSDLTVGQFYFLIRKRIHLRAEDALFFFVNNVIPPTSATMGQLYQEHHEEDFFLYIAYSDESVYGL