Reaction Details
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Report a problem with these dataTarget
Somatostatin receptor type 4
Ligand
BDBM81766
Substrate
n/a
Ki
1000±n/a nM
Comments
PDSP_1242
Citation
Hoyer, D; Lübbert, H; Bruns, C Molecular pharmacology of somatostatin receptors. Naunyn Schmiedebergs Arch Pharmacol 350:441-53 (1994) [PubMed] Article More Info.:
Target
Name:
Somatostatin receptor type 4
Synonyms:
SS-4-R | SS4-R | SS4R | SSR4_MOUSE | Smstr4 | Sstr4
Type:
PROTEIN
Mol. Mass.:
41937.48
Organism:
Mus musculus
Description:
ChEMBL_833920
Residue:
385
Sequence:
MNAPATLPPGVEDTTWTPGINASWAPDEEEEDAMGSDGTGTAGMVTIQCIYALVCLVGLVGNALVIFVILRYAKMKTATNIYLLNLAVADELFMLSVPFARSAAALRHWPFGAVLCRAVLSVDGLNMFTSVFCLTVLSVDRYVAVVHPLATATYRRPSVAKLINLGVWLASLLVTLPIAVFADTRPARGGEAVACNLHWPHPAWSAVFVIYTFLLGFLPPVLAIGLCYLLIVGKMRAVALAGGWQQRRRSEKKITRLVLMVVTVFVLCWMPFYVVQLLNLFVTSLDATVNHVSLILSYANSCANPILYGFLSDNFRRSFQRVLCLRCCLLETTGGAEEEPLDYYATALKSRGGAGCICPPLPCQQEPVQAEPGCKQVPFTKTTTF
Inhibitor
Name:
BDBM81766
Synonyms:
CAS_3086456 | MK 678 | NSC_3086456
Type:
Small organic molecule
Emp. Form.:
C44H56N8O7
Mol. Mass.:
808.9648
SMILES:
CC(C)C1NC(=O)C(CCCCN)NC(=O)C(Cc2c[nH]c3ccccc23)NC(=O)C(Cc2ccc(O)cc2)NC(=O)C(C)N(C)C(=O)C(Cc2ccccc2)NC1=O
Structure:
