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Reaction Details
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TargetPlatelet activating factor receptor
LigandBDBM50005240
Substrate/Competitorn/a
Meas. Tech.ChEBML_164926
IC50 690±n/a nM
Citation Carceller, EMerlos, MGiral, MBartrolí, JGarcía-Rafanell, JForn, J 4-substituted 2-alkoxytetrahydrofurans as potent and long-lasting PAF antagonists. J Med Chem35:676-83 (1992) [PubMed]  Article
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Platelet activating factor receptor
Name:Platelet activating factor receptor
Synonyms:PAF-R | Platelet-activating factor receptor
Type:Protein
Mol. Mass.:39005.63
Organism:Cavia porcellus
Description:n/a
Residue:342
Sequence:
MELNSSSRVDSEFRYTLFPIVYSIIFVLGIIANGYVLWVFARLYPSKKLNEIKIFMVNLT
VADLLFLITLPLWIVYYSNQGNWFLPKFLCNLAGCLFFINTYCSVAFLGVITYNRFQAVK
YPIKTAQATTRKRGIALSLVIWVAIVAAASYFLVMDSTNVVSNKAGSGNITRCFEHYEKG
SKPVLIIHICIVLGFFIVFLLILFCNLVIIHTLLRQPVKQQRNAEVRRRALWMVCTVLAV
FVICFVPHHMVQLPWTLAELGMWPSSNHQAINDAHQVTLCLLSTNCVLDPVIYCFLTKKF
RKHLSEKLNIMRSSQKCSRVTTDTGTEMAIPINHTPVNPIKN
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  Blast E-value cutoff:
BDBM50005240
NameBDBM50005240
Synonyms:2-({Acetyl-[5-(3-methyl-butoxy)-tetrahydro-furan-3-ylmethoxycarbonyl]-amino}-methyl)-1-ethyl-pyridinium; iodide | CHEMBL161674
TypeSmall organic molecule
Emp. Form.C21H33N2O5
Mol. Mass.393.4966
SMILESCC[n+]1ccccc1CN(C(C)=O)C(=O)OCC1COC(C1)OCCC(C)C
Structure
Search PDB for entries with ligand similarity:Similarity to this molecule at least:
n/a