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Reaction Details
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TargetPlatelet activating factor receptor
LigandBDBM50005228
Substrate/Competitorn/a
Meas. Tech.ChEBML_164926
IC50 51±n/a nM
Citation Carceller, EMerlos, MGiral, MBartrolí, JGarcía-Rafanell, JForn, J 4-substituted 2-alkoxytetrahydrofurans as potent and long-lasting PAF antagonists. J Med Chem35:676-83 (1992) [PubMed]  Article
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Platelet activating factor receptor
Name:Platelet activating factor receptor
Synonyms:PAF-R | Platelet-activating factor receptor
Type:Protein
Mol. Mass.:39005.63
Organism:Cavia porcellus
Description:n/a
Residue:342
Sequence:
MELNSSSRVDSEFRYTLFPIVYSIIFVLGIIANGYVLWVFARLYPSKKLNEIKIFMVNLT
VADLLFLITLPLWIVYYSNQGNWFLPKFLCNLAGCLFFINTYCSVAFLGVITYNRFQAVK
YPIKTAQATTRKRGIALSLVIWVAIVAAASYFLVMDSTNVVSNKAGSGNITRCFEHYEKG
SKPVLIIHICIVLGFFIVFLLILFCNLVIIHTLLRQPVKQQRNAEVRRRALWMVCTVLAV
FVICFVPHHMVQLPWTLAELGMWPSSNHQAINDAHQVTLCLLSTNCVLDPVIYCFLTKKF
RKHLSEKLNIMRSSQKCSRVTTDTGTEMAIPINHTPVNPIKN
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50005228
NameBDBM50005228
Synonyms:2-[(Acetyl-{5-[6-(3-phenyl-propoxy)-hexyloxy]-tetrahydro-furan-3-ylmethoxycarbonyl}-amino)-methyl]-1-ethyl-pyridinium; iodide | CHEMBL162251
TypeSmall organic molecule
Emp. Form.C31H45N2O6
Mol. Mass.541.6983
SMILESCC[n+]1ccccc1CN(C(C)=O)C(=O)OCC1COC(C1)OCCCCCCOCCCc1ccccc1
Structure
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n/a