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Target
Mu-type opioid receptor
Ligand
BDBM50000267
Substrate
n/a
Meas. Tech.
ChEMBL_145288 (CHEMBL752957)
Ki
3050±n/a nM
Citation
 Vecchietti, V; Giordani, A; Giardina, G; Colle, R; Clarke, GD (2S)-1-(arylacetyl)-2-(aminomethyl)piperidine derivatives: novel, highly selective kappa opioid analgesics. J Med Chem 34:397-403 (1991) [PubMed]  Article 
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:
Enzyme Catalytic Domain
Mol. Mass.:
11165.58
Organism:
GUINEA PIG
Description:
P97266
Residue:
98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
  
Inhibitor
Name:
BDBM50000267
Synonyms:
2-(3,4-Dichloro-phenyl)-1-(2-dimethylaminomethyl-piperidin-1-yl)-ethanone | 2-(3,4-Dichloro-phenyl)-1-(2-dimethylaminomethyl-piperidin-1-yl)-ethanone(HCl) | CHEMBL339552
Type:
Small organic molecule
Emp. Form.:
C16H22Cl2N2O
Mol. Mass.:
329.265
SMILES:
CN(C)CC1CCCCN1C(=O)Cc1ccc(Cl)c(Cl)c1
Structure:
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