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TargetAGTR1
LigandBDBM50082569
Substrate/Competitorn/a
Meas. Tech.ChEMBL_35127
Ki 22±n/a nM
Citation Nouet, SDodey, PRBondoux, MRPruneau, DLuccarini, JMGroblewski, TLarguier, RLombard, CMarie, JRenaut, PPLeclerc, GBonnafous, JC Specific nonpeptide photoprobes as tools for the structural study of the angiotensin II AT(1) receptor. J Med Chem42:4572-83 (1999) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
AGTR1
Name:AGTR1
Synonyms:ANGIOTENSIN AT1 | Angiotensin II AT1 | Angiotensin II AT1A | Angiotensin II receptor (AT-1) type-1 | Type-1A angiotensin II receptor
Type:Enzyme Catalytic Domain
Mol. Mass.:40910.53
Organism:RAT
Description:ANGIOTENSIN AT1 AGTR1 RAT::P25095
Residue:359
Sequence:
MALNSSAEDGIKRIQDDCPKAGRHSYIFVMIPTLYSIIFVVGIFGNSLVVIVIYFYMKLK
TVASVFLLNLALADLCFLLTLPLWAVYTAMEYRWPFGNHLCKIASASVSFNLYASVFLLT
CLSIDRYLAIVHPMKSRLRRTMLVAKVTCIIIWLMAGLASLPAVIHRNVYFIENTNITVC
AFHYESRNSTLPIGLGLTKNILGFLFPFLIILTSYTLIWKALKKAYEIQKNKPRNDDIFR
IIMAIVLFFFFSWVPHQIFTFLDVLIQLGVIHDCKISDIVDTAMPITICIAYFNNCLNPL
FYGFLGKKFKKYFLQLLKYIPPKAKSHSSLSTKMSTLSYRPSDNMSSSAKKPASCFEVE
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  Blast E-value cutoff:
BDBM50082569
n/a
NameBDBM50082569
Synonyms:4-Azido-2-{[2-butyl-3-(4-carboxy-benzyl)-3H-imidazol-4-ylmethyl]-amino}-benzoic acid | 4-azido-2-[2-butyl-1-(4-carboxybenzyl)-1H-5-imidazolylmethylamino]benzoic acid | CHEMBL141065
TypeSmall organic molecule
Emp. Form.C23H24N6O4
Mol. Mass.448.4745
SMILESCCCCc1ncc(CNc2cc(ccc2C(O)=O)N=[N+]=[N-])n1Cc1ccc(cc1)C(O)=O
Structure
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