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Target
Delta-type opioid receptor
Ligand
BDBM50083735
Substrate
n/a
Meas. Tech.
ChEBML_53451
IC50
9327±n/a nM
Citation
 Burden, JE; Davis, P; Porreca, F; Spatola, AF Synthesis and biological activities of position one and three transposed analogs of the opioid peptide YKFA. Bioorg Med Chem Lett 9:3441-6 (2000) [PubMed]  Article 
Target
Name:
Delta-type opioid receptor
Synonyms:
DOR-1 | K56 | MSL-2 | OPIATE Delta | OPRD_MOUSE | Opioid receptors; mu and delta | Oprd1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
40577.25
Organism:
MOUSE
Description:
P32300
Residue:
372
Sequence:
MELVPSARAELQSSPLVNLSDAFPSAFPSAGANASGSPGARSASSLALAIAITALYSAVCAVGLLGNVLVMFGIVRYTKLKTATNIYIFNLALADALATSTLPFQSAKYLMETWPFGELLCKAVLSIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGVGVPIMVMAVTQPRDGAVVCMLQFPSPSWYWDTVTKICVFLFAFVVPILIITVCYGLMLLRLRSVRLLSGSKEKDRSLRRITRMVLVVVGAFVVCWAPIHIFVIVWTLVDINRRDPLVVAALHLCIALGYANSSLNPVLYAFLDENFKRCFRQLCRTPCGRQEPGSLRRPRQATTRERVTACTPSDGPGGGAAA
  
Inhibitor
Name:
BDBM50083735
Synonyms:
(R)-2-Amino-N-[(R)-6-(4-hydroxy-benzyl)-3-methyl-2,5,8-trioxo-1,4,7triaza-cyclotridec-9-yl]-3-phenyl-propionamide | CHEMBL2370484
Type:
Small organic molecule
Emp. Form.:
C27H35N5O5
Mol. Mass.:
509.5973
SMILES:
C[C@@H]1NC(=O)[C@H](Cc2ccc(O)cc2)NC(=O)[C@@H](CCCCNC1=O)NC(=O)[C@H](N)Cc1ccccc1
Structure:
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