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TargetBeta tubulin
LigandBDBM50012278
Substrate/Competitorn/a
Meas. Tech.ChEMBL_311916
IC50 1000±n/a nM
Citation Morita, HKoyama, KSugimoto, YKobayashi, J Antimitotic activity and reversal of breast cancer resistance protein-mediated drug resistance by stilbenoids from Bletilla striata. Bioorg Med Chem Lett15:1051-4 (2005) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Beta tubulin
Name:Beta tubulin
Synonyms:n/a
Type:PROTEIN
Mol. Mass.:4652.47
Organism:Leishmania donovani
Description:ChEMBL_311916
Residue:43
Sequence:
MREIVSCQAGQCGNQIGSKFWEVIADEHGVDPTGSYQGDSDLQ
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  Blast E-value cutoff:
BDBM50012278
NameBDBM50012278
Synonyms:(2ALPHA,2''BETA,3BETA,4ALPHA,5BETA)-VINCALEUKOBLASTINE | CHEMBL159 | VINBLASTINE | VINBLASTINE SULFATE | cid_5388983
TypeSmall organic molecule
Emp. Form.C46H58N4O9
Mol. Mass.810.9741
SMILESCC[C@]1(O)C[C@@H]2CN(C1)CCc1c([nH]c3ccccc13)[C@@](C2)(C(=O)OC)c1cc2c(cc1OC)N(C)[C@@H]1[C@]22CCN3CC=C[C@](CC)([C@@H]23)[C@@H](OC(C)=O)[C@]1(O)C(=O)OC |r,c:48|
Structure
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