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TargetPurinergic receptor P2Y14
LigandBDBM50209663
Substrate/Competitorn/a
Meas. Tech.ChEMBL_434326
EC50 350±n/a nM
Citation Ko, HFricks, IIvanov, AAHarden, TKJacobson, KA Structure-activity relationship of uridine 5'-diphosphoglucose analogues as agonists of the human P2Y14 receptor. J Med Chem50:2030-9 (2007) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Purinergic receptor P2Y14
Name:Purinergic receptor P2Y14
Synonyms:n/a
Type:PROTEIN
Mol. Mass.:38991.62
Organism:Homo sapiens (Human)
Description:ChEMBL_1502487
Residue:338
Sequence:
MINSTSTQPPDESCSQNLLITQQIIPVLYCMVFIAGILLNGVSGWIFFYVPSSKSFIIYL
KNIVIADFVMSLTFPFKILGDSGLGPWQLNVFVCRVSAVLFYVNMYVSIVFFGLISFDRY
YKIVKPLWTSFIQSVSYSKLLSVIVWMLMLLLAVPNIILTNQSVREVTQIKCIELKSELG
RKWHKASNYIFVAIFWIVFLLLIVFYTAITKKIFKSHLKSSRNSTSVKKKSSRNIFSIVF
VFFVCFVPYHIARIPYTKSQTEAHYSCQSKEILRYMKEFTLLLSAANVCLDPIIYFFLCQ
PFREILCKKLHIPLKAQNDLDISRIKRGNTTLESTDTL
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BDBM50209663
NameBDBM50209663
Synonyms:CHEMBL374384 | MRS-2670 | diphosphoric acid 1-alpha-D-glucopyranosyl ester 2-((4'-thio)uridin-5''-yl) ester
TypeSmall organic molecule
Emp. Form.C15H24N2O16P2S
Mol. Mass.582.367
SMILESOC[C@H]1O[C@H](OP(O)(=O)OP(O)(=O)OC[C@H]2O[C@H]([C@H](O)[C@@H]2O)n2ccc(=S)[nH]c2=O)[C@H](O)[C@@H](O)[C@@H]1O
Structure
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n/a