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Target
Protein ADM2
Ligand
BDBM50246697
Substrate
n/a
Meas. Tech.
ChEMBL_556927 (CHEMBL954953)
IC50
318±n/a nM
Citation
 Miranda, LP; Holder, JR; Shi, L; Bennett, B; Aral, J; Gegg, CV; Wright, M; Walker, K; Doellgast, G; Rogers, R; Li, H; Valladares, V; Salyers, K; Johnson, E; Wild, K Identification of potent, selective, and metabolically stable peptide antagonists to the calcitonin gene-related peptide (CGRP) receptor. J Med Chem 51:7889-97 (2008) [PubMed]  Article 
Target
Name:
Protein ADM2
Synonyms:
ADM2 | ADM2_HUMAN | AM2
Type:
PROTEIN
Mol. Mass.:
15883.28
Organism:
Homo sapiens (Human)
Description:
ChEMBL_556927
Residue:
148
Sequence:
MARIPTAALGCISLLCLQLPGSLSRSLGGDPRPVKPREPPARSPSSSLQPRHPAPRPVVWKLHRALQAQRGAGLAPVMGQPLRDGGRQHSGPRRHSGPRRTQAQLLRVGCVLGTCQVQNLSHRLWQLMGPAGRQDSAPVDPSSPHSYG
  
Inhibitor
Name:
BDBM50246697
Synonyms:
Ac-WVTH[Cit]LAGLLS[Cit]SGGVV[hArg]KNFVPTDVGPFAF-NH2 | CHEMBL525039
Type:
Small organic molecule
Emp. Form.:
C160H246N44O41
Mol. Mass.:
3441.9354
SMILES:
n/a
Structure:
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