Reaction Details Report a problem with these data
Target
Transcription factor Jun
Ligand
BDBM50326017
Substrate
n/a
Meas. Tech.
ChEMBL_654663 (CHEMBL1243707)
Kd
10000±n/a nM
Citation
 Luedtke, NW; Dexter, RJ; Fried, DB; Schepartz, A Surveying polypeptide and protein domain conformation and association with FlAsH and ReAsH. Nat Chem Biol 3:779-84 (2007) [PubMed]  Article 
Target
Name:
Transcription factor Jun
Synonyms:
AP1 | Activator protein 1 | JUN | JUN_HUMAN | Proto-oncogene c-JUN | Transcription factor AP-1 | Transcription factor AP1 | V-jun avian sarcoma virus 17 oncogene homolog | p39
Type:
n/a
Mol. Mass.:
35683.24
Organism:
Homo sapiens (Human)
Description:
P05412
Residue:
331
Sequence:
MTAKMETTFYDDALNASFLPSESGPYGYSNPKILKQSMTLNLADPVGSLKPHLRAKNSDLLTSPDVGLLKLASPELERLIIQSSNGHITTTPTPTQFLCPKNVTDEQEGFAEGFVRALAELHSQNTLPSVTSAAQPVNGAGMVAPAVASVAGGSGSGGFSASLHSEPPVYANLSNFNPGALSSGGGAPSYGAAGLAFPAQPQQQQQPPHHLPQQMPVQHPRLQALKEEPQTVPEMPGETPPLSPIDMESQERIKAERKRMRNRIAASKCRKRKLERIARLEEKVKTLKAQNSELASTANMLREQVAQLKQKVMNHVNSGCQLMLTQQLQTF
  
Inhibitor
Name:
BDBM50326017
Synonyms:
Ac-WRIARLEEKVKTLKAQNSELASTANMLREQVAQLKQKVCC-NH2 | CHEMBL1241036
Type:
Small organic molecule
Emp. Form.:
C200H344N62O59S3
Mol. Mass.:
4657.446
SMILES:
n/a
Structure:
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