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Target
Beta-lactamase
Ligand
BDBM50021959
Substrate
n/a
Meas. Tech.
ChEMBL_703757 (CHEMBL1657725)
IC50
235520±n/a nM
Citation
Beceiro, A; Pérez, A; Fernández-Cuenca, F; Martínez-Martínez, L; Pascual, A; Vila, J; Rodríguez-Baño, J; Cisneros, JM; Pachón, J; Bou, G Genetic variability among ampC genes from acinetobacter genomic species 3. Antimicrob Agents Chemother 53:1177-84 (2009) [PubMed] Article
More Info.:
Target
Name:
Beta-lactamase
Synonyms:
ADC-14 protein
Type:
PROTEIN
Mol. Mass.:
43128.73
Organism:
Acinetobacter genomosp. 3
Description:
ChEMBL_703757
Residue:
383
Sequence:
MRFKKISCLLLSPLFIFSTSIYAGNTPKDQEIKKLVDQNFKPLLEKYDVPGMAVGVIQNNKKYEIYYGLQSVQDKKAVNSSTIFELGSVSKLFTATAGGYAKTKGTISFKDTPGKYWKELKNTPIDQVNLLQLATYTSGNLALQFPDEVQTDQQVLTFFKDWKPKNPIGEYRQYSNPSIGLFGKVVALSMNKPFDQVLEKTIFPGLSLKHSYVNVPKTQMQNYAFGYNQENQPIRVNPGPLDAPAYGVKSTLPDMLKFINANLNPQKYPADIQRAINETHQGFYQVGTMYQALGWEEFSYPAPLQTLLDSNSEQIVMKPNKVTAISKEPSVKMFHKTGSTNGFGTYVVFIPKENIGLVMLTNKRIPNEERFKAAYAVLNAIKK