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Target
Calmodulin-1
Ligand
BDBM50346807
Substrate
n/a
Meas. Tech.
ChEMBL_753876 (CHEMBL1798138)
IC50
62680±n/a nM
Citation
Reyes-Ramírez, A; Leyte-Lugo, M; Figueroa, M; Serrano-Alba, T; González-Andrade, M; Mata, R Synthesis, biological evaluation, and docking studies of gigantol analogs as calmodulin inhibitors. Eur J Med Chem 46:2699-708 (2011) [PubMed] Article
More Info.:
Target
Name:
Calmodulin-1
Synonyms:
CALM | CALM1 | CALM1_HUMAN | CALM2 | CAM | CAM1 | CAM2 | CAMB | Calmodulin-2
Type:
Protein
Mol. Mass.:
16813.73
Organism:
Human
Description:
P0DP23
Residue:
149
Sequence:
MADQLTEEQIAEFKEAFSLFDKDGDGTITTKELGTVMRSLGQNPTEAELQDMINEVDADGNGTIDFPEFLTMMARKMKDTDSEEEIREAFRVFDKDGNGYISAAELRHVMTNLGEKLTDEEVDEMIREADIDGDGQVNYEEFVQMMTAK