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Reaction Details
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TargetTrace amine-associated receptor 1 (TAAR1)
LigandBDBM50359505
Substrate/Competitorn/a
Meas. Tech.ChEMBL_792739
EC50 22.4±n/a nM
Citation Lewin, AHMiller, GMGilmour, B Trace amine-associated receptor 1 is a stereoselective binding site for compounds in the amphetamine class. Bioorg Med Chem19:7044-8 (2011) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Trace amine-associated receptor 1 (TAAR1)
Name:Trace amine-associated receptor 1
Synonyms:Trace amine receptor 1 (TARR1) | Trace amine-associated receptor1
Type:Enzyme
Mol. Mass.:38034.73
Organism:Rattus norvegicus (Rat)
Description:Q923Y9
Residue:332
Sequence:
MHLCHNSANISHTNSNWSRDVRASLYSLISLIILTTLVGNLIVIISISHFKQLHTPTNWL
LHSMAVVDFLLGCLVMPYSMVRTVEHCWYFGELFCKLHTSTDIMLSSASILHLAFISIDR
YYAVCDPLRYKAKINLAAIFVMILISWSLPAVFAFGMIFLELNLEGVEELYHNQVFCLRG
CFPFFSKVSGVLAFMTSFYIPGSVMLFVYYRIYFIAKGQARSINRANLQVGLEGESRAPQ
SKETKAAKTLGIMVGVFLLCWCPFFFCMVLDPFLGYVIPPTLNDTLNWFGYLNSAFNPMV
YAFFYPWFRRALKMVLFGKIFQKDSSRSKLFL
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  Blast E-value cutoff:
BDBM50359505
NameBDBM50359505
Synonyms:CHEMBL1182312
TypeSmall organic molecule
Emp. Form.C14H14INO2
Mol. Mass.355.1709
SMILESNCCc1ccc(Oc2ccc(O)cc2)c(I)c1
Structure
Search PDB for entries with ligand similarity:Similarity to this molecule at least:
n/a